SCHEMBL21452841

SCHEMBL21452841

C/C=C\Cc1ccc(C(F)(F)F)c(C)c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.44
IDO1 P14902 4/20 0.37
PDE2A O00408 2/20 0.34
FFAR4 Q5NUL3 2/20 0.33
KIF11 P52732 2/20 0.33
FFAR1 O14842 1/20 0.33
FAAH O00519 1/20 0.33
MGLL Q99685 1/20 0.33
SIGMAR1 Q99720 1/20 0.32
RXRA P19793 1/20 0.32
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32
OPRK1 P41145 1/20 0.31
AKR1C4 P17516 2/20 0.30
AKR1C3 P42330 2/20 0.30
AKR1C2 P52895 2/20 0.30
RAPGEF4 Q8WZA2 1/20 0.30
AKR1C1 Q04828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4593166 0.81 DAO (0.50) DAOPDE2AFFAR4KIF11FFAR1
SCHEMBL15385131 0.79 DAO (0.48) DAOIDO1PDE2AKIF11
SCHEMBL590101 0.79 ALDH1A1 (0.39) AKR1C4AKR1C3AKR1C2AKR1C1
SCHEMBL22296720 0.79 GLA (0.37) IDO1PDE2A
Hydrochloric Acid SCHEMBL23165936 0.78 DAO (0.47) DAOIDO1PDE2AKIF11
SCHEMBL12886693 0.77 PDE2A (0.53) DAOIDO1PDE2AFFAR4KIF11
SCHEMBL13598345 0.76 DAO (0.48) DAOIDO1PDE2AFFAR4KIF11
SCHEMBL29277330 0.76 DAO (0.48) DAOIDO1PDE2AFFAR4KIF11
SCHEMBL3901935 0.76 KIF11 (0.51) DAOPDE2AFFAR4KIF11FFAR1
SCHEMBL11618144 0.75 DAO (0.44) DAOIDO1PDE2AKIF11RAPGEF4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019193516-A2 SUBSTITUTED PYRIDINE AND PYRIMIDINES AND THEIR USE AS GLUN2B RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2019-10-10 WO disclosed