SCHEMBL21456788

SCHEMBL21456788

CC(C)(O)C(C)(C)O.O=S(=O)(c1ccccc1)n1ccc2c(B(O)O)ccnc21

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.49
HTR6 P50406 11/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
MET P08581 1/20 0.40
PIK3C3 Q8NEB9 3/20 0.40
PKM P14618 1/20 0.38
HTR1A P08908 1/20 0.37
DRD2 P14416 1/20 0.37
HTR2A P28223 1/20 0.37
ENPP3 O14638 1/20 0.36
ENPP1 P22413 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29952621 0.94 CYP2C19 (0.55) CYP2C19HTR6L3MBTL1METPIK3C3
SCHEMBL18155085 0.87 CYP2C19 (0.44) CYP2C19HTR6L3MBTL1METPIK3C3
SCHEMBL12272025 0.83 L3MBTL1 (0.56) CYP2C19HTR6L3MBTL1PKM
SCHEMBL1672537 0.77 CYP2C19 (0.58) CYP2C19HTR6L3MBTL1METPKM
SCHEMBL17394567 0.76 HTR6 (0.58) CYP2C19HTR6L3MBTL1MET
SCHEMBL21821845 0.75 CYP2C19 (0.56) CYP2C19HTR6L3MBTL1METPKM
SCHEMBL16516498 0.74 HTR6 (0.50) CYP2C19HTR6L3MBTL1METPKM
SCHEMBL1683430 0.74 CYP2C19 (0.58) CYP2C19HTR6L3MBTL1METPKM
SCHEMBL457569 0.74 CYP2C19 (0.58) CYP2C19HTR6L3MBTL1METPKM
SCHEMBL414843 0.74 CYP2C19 (0.58) CYP2C19HTR6L3MBTL1METPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3283475-B1 3-(1H-BENZIMIDAZOL-2-YL)-1H-PYRIDIN-2-ONE DERIVATIVES MERCK PATENT GMBH (DE) 2019-10-16 EP disclosed