SCHEMBL2146384

SCHEMBL2146384

O=C(O)N1CC(O)C(Oc2ccccc2F)C1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 2/20 0.39
GRIN2B Q13224 2/20 0.39
HPGD P15428 2/20 0.39
RIPK1 Q13546 1/20 0.38
FKBP1A P62942 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CXCL8 P10145 1/20 0.36
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KDM4E B2RXH2 1/20 0.35
LPAR1 Q92633 1/20 0.35
LPAR5 Q9H1C0 1/20 0.35
PPARG P37231 1/20 0.35
PPARA Q07869 1/20 0.35
NOTUM Q6P988 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2146128 0.86 GRIN1 (0.41) GRIN1GRIN2BHPGDL3MBTL1ALDH1A1
SCHEMBL2146132 0.79 GAA (0.40) GRIN1GRIN2BFKBP1AALDH1A1MAPT
SCHEMBL28383178 0.77 GRIN2B (0.58) GRIN1GRIN2BRIPK1
SCHEMBL17633359 0.77 GRIN2B (0.58) GRIN1GRIN2BRIPK1
SCHEMBL17633278 0.77 GRIN2B (0.58) GRIN1GRIN2BRIPK1
SCHEMBL17633280 0.77 GRIN2B (0.58) GRIN1GRIN2BRIPK1
SCHEMBL2146215 0.75 MEN1 (0.42) ALDH1A1PPARGPPARA
SCHEMBL27076325 0.75 GRIN1 (0.36) GRIN1GRIN2BHPGDRIPK1FKBP1A
SCHEMBL27076326 0.75 GRIN1 (0.36) GRIN1GRIN2BHPGDRIPK1FKBP1A
SCHEMBL27076333 0.75 GRIN1 (0.36) GRIN1GRIN2BHPGDRIPK1FKBP1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011088045-A1 AURORA KINASE COMPOUNDS AND METHODS OF THEIR USE AMBIT BIOSCIENCES CORPORATION (US) 2011-07-21 WO disclosed