SCHEMBL2146128

SCHEMBL2146128

O=C(O)N1CC(O)C(Oc2ccc(F)cc2F)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 3/20 0.41
GRIN2B Q13224 3/20 0.41
RBP4 P02753 2/20 0.37
MKNK2 Q9HBH9 2/20 0.37
GPR6 P46095 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
SCN9A Q15858 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CPS1 P31327 2/20 0.34
POLB P06746 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2146384 0.86 GRIN1 (0.39) GRIN1GRIN2BALDH1A1MAPTHPGD
SCHEMBL2146132 0.80 GAA (0.40) GRIN1GRIN2BALDH1A1LMNAMEN1
SCHEMBL2146215 0.78 MEN1 (0.42) ALDH1A1MEN1KMT2A
SCHEMBL27900160 0.76 MGLL (0.40) NPC1RAB9A
SCHEMBL12497264 0.74 TRPV4 (0.44) SCN9AHPGD
SCHEMBL16801543 0.73 MKNK2 (0.47) MKNK2GPR6
SCHEMBL16801870 0.73 MKNK2 (0.47) MKNK2GPR6
SCHEMBL18982966 0.73 MKNK2 (0.47) MKNK2GPR6
SCHEMBL4199136 0.73 ALDH1A1 (0.41) ALDH1A1LMNATDP1MEN1KMT2A
SCHEMBL19006122 0.70 MKNK2 (0.45) MKNK2GPR6ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011088045-A1 AURORA KINASE COMPOUNDS AND METHODS OF THEIR USE AMBIT BIOSCIENCES CORPORATION (US) 2011-07-21 WO disclosed