SCHEMBL2146789

SCHEMBL2146789

O[C@@H]1CNC[C@@H]1Oc1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.38
SLC6A2 P23975 2/20 0.35
NPY1R P25929 1/20 0.35
NPY2R P49146 1/20 0.35
NPY4R P50391 1/20 0.35
NPY5R Q15761 1/20 0.35
LTA4H P09960 1/20 0.35
PTPN2 P17706 2/20 0.35
PTPN1 P18031 2/20 0.35
PTPN11 Q06124 2/20 0.35
MAN1B1 Q9UKM7 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
LMNA P02545 1/20 0.34
EPHX2 P34913 1/20 0.34
MKNK2 Q9HBH9 2/20 0.34
GRK2 P25098 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2146784 1.00 TRPA1 (0.38) TRPA1SLC6A2NPY1RNPY2RNPY4R
SCHEMBL2146780 1.00 TRPA1 (0.38) TRPA1SLC6A2NPY1RNPY2RNPY4R
SCHEMBL11244532 0.85 HTR2B (0.42) TRPA1SLC6A2NPY1RNPY2RNPY4R
SCHEMBL11244526 0.85 HTR2B (0.42) TRPA1SLC6A2NPY1RNPY2RNPY4R
SCHEMBL11236259 0.85 HTR2B (0.42) TRPA1SLC6A2NPY1RNPY2RNPY4R
SCHEMBL11236271 0.85 HTR2B (0.42) TRPA1SLC6A2NPY1RNPY2RNPY4R
SCHEMBL11236266 0.85 HTR2B (0.42) TRPA1SLC6A2NPY1RNPY2RNPY4R
SCHEMBL10839532 0.84 MEN1 (0.37) SLC6A2NPY1RNPY2RNPY4RNPY5R
SCHEMBL10839525 0.84 MEN1 (0.37) SLC6A2NPY1RNPY2RNPY4RNPY5R
SCHEMBL10839528 0.84 MEN1 (0.37) SLC6A2NPY1RNPY2RNPY4RNPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011088045-A1 AURORA KINASE COMPOUNDS AND METHODS OF THEIR USE AMBIT BIOSCIENCES CORPORATION (US) 2011-07-21 WO disclosed