SCHEMBL21468656

SCHEMBL21468656

Cn1ccc(OC[Si](C)(C)C)n1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.38
CYP19A1 P11511 1/20 0.38
KMT2A Q03164 1/20 0.35
KEAP1 Q14145 1/20 0.33
SIGMAR1 Q99720 5/20 0.33
EPHX2 P34913 1/20 0.33
JMJD6 Q6NYC1 3/20 0.32
SCN4A P35499 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
DDB1 Q16531 1/20 0.31
CRBN Q96SW2 1/20 0.31
TSHR P16473 1/20 0.31
ABL1 P00519 1/20 0.31
NOTUM Q6P988 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2629335 0.79
SCHEMBL7810321 0.78
SCHEMBL21468722 0.77 DYRK1A (0.37)
SCHEMBL18222561 0.74 CYP19A1 (0.40) KDM1ACYP19A1KMT2AKEAP1SIGMAR1
SCHEMBL17662643 0.74 JMJD6 (0.43) KDM1ACYP19A1KMT2AKEAP1SIGMAR1
SCHEMBL18222497 0.74 CYP19A1 (0.44) KDM1ACYP19A1KMT2AKEAP1SIGMAR1
SCHEMBL21438893 0.73 HTT (0.32) ALDH1A1HTTSMN1; SMN2
SCHEMBL9384706 0.72 TDP1 (0.41) KDM1ACYP19A1EPHX2JMJD6HTT
SCHEMBL12970421 0.72 PKM (0.59) KDM1AKMT2AEPHX2JMJD6SMN1; SMN2
SCHEMBL19121810 0.72 CYP19A1 (0.38) KDM1ACYP19A1KMT2AKEAP1JMJD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019200246-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR, PHARMACEUTICAL COMPOSITIONS, METHODS OF TREATMENT, AND PROCESS FOR MAKING THE MODULATOR ABELA ALEXANDER RUSSELL (US) 2019-10-17 WO disclosed