SCHEMBL21473669

SCHEMBL21473669

CNC(=O)C(c1ccccc1)N1Cc2ccccc2C1=O

nearest known ligand 0.79

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
THRB P10828 5/20 0.79
KDM4E B2RXH2 1/20 0.72
ALDH1A1 P00352 1/20 0.72
ALOX15 P16050 1/20 0.72
TSHR P16473 1/20 0.72
XIAP P98170 1/20 0.72
HKDC1 Q2TB90 1/20 0.72
HSD17B10 Q99714 1/20 0.72
TDP1 Q9NUW8 1/20 0.72
L3MBTL1 Q9Y468 1/20 0.72
MAPT P10636 2/20 0.67
LMNA P02545 2/20 0.65
EGFR P00533 1/20 0.63
GAA P10253 2/20 0.62
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
SDCBP O00560 1/20 0.54
SDC2 P34741 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22997167 1.00 THRB (0.79) THRBKDM4EALDH1A1ALOX15TSHR
SCHEMBL18360800 0.88 THRB (0.84) THRBKDM4EALDH1A1ALOX15TSHR
SCHEMBL20527883 0.88 THRB (0.84) THRBKDM4EALDH1A1ALOX15TSHR
SCHEMBL21473573 0.88 THRB (1.00) THRBKDM4EALDH1A1ALOX15TSHR
SCHEMBL18360734 0.87 THRB (0.83) THRBKDM4EALDH1A1ALOX15TSHR
SCHEMBL20527801 0.87 THRB (0.83) THRBKDM4EALDH1A1ALOX15TSHR
SCHEMBL18360735 0.87 THRB (0.83) THRBKDM4EALDH1A1ALOX15TSHR
SCHEMBL20527800 0.87 THRB (0.83) THRBKDM4EALDH1A1ALOX15TSHR
SCHEMBL20527890 0.87 THRB (0.83) THRBKDM4EALDH1A1ALOX15TSHR
SCHEMBL21473668 0.87 THRB (0.61) THRBKDM4EALDH1A1ALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020211853-A1 NOVEL EGFR TRIPLE MUTATION INHIBITOR AND APPLICATION THEREOF 华东理工大学 2020-10-22 WO disclosed
WO-2019196938-A1 QUINAZOLINE COMPOUND SERVING AS EGFR TRIPLE MUTATION INHIBITOR AND APPLICATIONS THEREOF 华东理工大学 2019-10-17 WO disclosed