SCHEMBL21473668

SCHEMBL21473668

CNC(=O)C(c1cccc(F)c1)N1Cc2ccccc2C1=O

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
THRB P10828 7/20 0.61
LMNA P02545 3/20 0.58
MAPT P10636 1/20 0.56
KDM4E B2RXH2 1/20 0.55
ALDH1A1 P00352 1/20 0.55
ALOX15 P16050 1/20 0.55
TSHR P16473 1/20 0.55
XIAP P98170 1/20 0.55
HKDC1 Q2TB90 1/20 0.55
HSD17B10 Q99714 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
EGFR P00533 3/20 0.50
GAA P10253 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23424771 0.88 THRB (0.57) THRBLMNAMAPTKDM4EALDH1A1
SCHEMBL22997167 0.87 THRB (0.79) THRBLMNAMAPTKDM4EALDH1A1
SCHEMBL21473669 0.87 THRB (0.79) THRBLMNAMAPTKDM4EALDH1A1
SCHEMBL23424769 0.86 THRB (0.55) THRBLMNAMAPTKDM4EALDH1A1
SCHEMBL30046742 0.85 ALOX15 (0.59) THRBLMNAMAPTKDM4EALDH1A1
SCHEMBL22997586 0.83 EGFR (0.56) THRBLMNAMAPTKDM4EALDH1A1
SCHEMBL20527835 0.77 THRB (0.65) THRBLMNAMAPTKDM4EALDH1A1
SCHEMBL18360811 0.77 THRB (0.65) THRBLMNAMAPTKDM4EALDH1A1
SCHEMBL21473592 0.76 MEN1 (0.55) THRBLMNAMAPTKDM4EALDH1A1
SCHEMBL20527883 0.76 THRB (0.84) THRBLMNAMAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019196938-A1 QUINAZOLINE COMPOUND SERVING AS EGFR TRIPLE MUTATION INHIBITOR AND APPLICATIONS THEREOF 华东理工大学 2019-10-17 WO disclosed