SCHEMBL2148563

SCHEMBL2148563

Cc1cc(Nc2nc(Sc3ccc(NC(=O)c4c(C(F)(F)F)nn(C)c4Cl)cc3)nc3cccn23)n[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.47
CYP3A4 P08684 3/20 0.47
CYP2C19 P33261 2/20 0.47
ALDH1A1 P00352 1/20 0.47
POLB P06746 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CYP2C9 P11712 2/20 0.45
AURKA O14965 14/20 0.43
AURKB Q96GD4 14/20 0.43
AURKC Q9UQB9 5/20 0.42
SRC P12931 2/20 0.41
GSK3B P49841 1/20 0.41
ABL1 P00519 2/20 0.41
BCR P11274 2/20 0.41
PLK4 O00444 2/20 0.41
BMPR1B O00238 1/20 0.41
STK25 O00506 1/20 0.41
RIOK3 O14730 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2149056 0.83 AURKB (0.44) AURKAAURKBAURKCSRCGSK3B
SCHEMBL2148756 0.82 AURKB (0.46) AURKAAURKBAURKCSRCGSK3B
SCHEMBL2948567 0.81 AURKB (0.64) AURKAAURKBAURKCSRCGSK3B
SCHEMBL2146309 0.80 AURKB (0.55) AURKAAURKBAURKCSRCGSK3B
SCHEMBL2169729 0.77 AURKB (0.65) AURKAAURKBAURKCSRCGSK3B
SCHEMBL2161109 0.76 AURKB (0.56) AURKAAURKBAURKCSRCGSK3B
SCHEMBL2148867 0.74 AURKA (0.47) AURKAAURKBAURKCSRCGSK3B
SCHEMBL2160263 0.74 AURKB (0.68) AURKAAURKBAURKCSRCGSK3B
SCHEMBL2148590 0.74 AURKA (0.55) AURKAAURKBAURKC
SCHEMBL2150067 0.74 AURKB (0.56) AURKAAURKBAURKC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011088045-A1 AURORA KINASE COMPOUNDS AND METHODS OF THEIR USE AMBIT BIOSCIENCES CORPORATION (US) 2011-07-21 WO disclosed