SCHEMBL21486341

SCHEMBL21486341

N/C=C/c1ccc(Oc2c(F)cccc2F)cc1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 8/20 0.40
RELA Q04206 3/20 0.40
LPAR1 Q92633 1/20 0.36
LPAR5 Q9H1C0 1/20 0.36
HTR1A P08908 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
KCNH2 Q12809 2/20 0.34
MAT2A P31153 1/20 0.34
DHODH Q02127 1/20 0.34
TLR4 O00206 1/20 0.33
TLR2 O60603 1/20 0.33
ESR1 P03372 1/20 0.33
PTGES2 Q9H7Z7 1/20 0.33
PARP10 Q53GL7 1/20 0.33
POLB P06746 1/20 0.33
HSP90AA1 P07900 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL505416 0.78 ALDH1A1 (0.50) LPAR1LPAR5DHODHPARP10POLB
SCHEMBL21483129 0.76 TLR4 (0.65) TLR4TLR2
SCHEMBL15515736 0.75 ALDH1A1 (0.54) LPAR1LPAR5POLBHSP90AA1MAPT
SCHEMBL21486338 0.71 TEAD4 (0.45) NFE2L2LPAR1LPAR5HTR1ASLC6A2
SCHEMBL17423587 0.71 MAPT (0.45) LPAR1LPAR5HTR1ASLC6A2SLC6A4
SCHEMBL13861391 0.71 LPAR1 (0.40) LPAR1LPAR5HTR1ASLC6A2SLC6A4
SCHEMBL1129355 0.71 MAPT (0.45) LPAR1LPAR5HTR1ASLC6A2SLC6A4
SCHEMBL5539624 0.71 LPAR1 (0.40) LPAR1LPAR5HTR1ASLC6A2SLC6A4
SCHEMBL23170416 0.70 HSD17B10 (0.41) LPAR1LPAR5HTR1ASLC6A2SLC6A4
SCHEMBL16415975 0.68 SLC6A2 (0.45) NFE2L2LPAR1LPAR5HTR1ASLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019196915-A1 METHOD FOR PREPARING PYRROLOAMINOPYRIDAZINONE COMPOUND AND INTERMEDIATES THEREOF 江苏恒瑞医药股份有限公司 2019-10-17 WO disclosed