SCHEMBL21486451

SCHEMBL21486451

CC(C)c1cnn2c(N)nc(N3CCC(N)CC3)nc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.37
HRH4 Q9H3N8 1/20 0.37
CDK2 P24941 13/20 0.37
GSK3B P49841 2/20 0.37
CDK9 P50750 10/20 0.36
CCNT1 O60563 3/20 0.35
CDK5 Q00535 3/20 0.35
CDK5R1 Q15078 3/20 0.35
CCNA2 P20248 2/20 0.35
DYRK3 O43781 1/20 0.35
CLK1 P49759 1/20 0.35
CLK2 P49760 1/20 0.35
CLK3 P49761 1/20 0.35
DYRK1A Q13627 1/20 0.35
DYRK2 Q92630 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
DYRK1B Q9Y463 1/20 0.35
PAK1 Q13153 1/20 0.34
PTPN11 Q06124 1/20 0.33
PAK4 O96013 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26973963 0.87 CDK2 (0.37) HRH3HRH4CDK2GSK3BCDK9
SCHEMBL21481495 0.82 CDK2 (0.36) CDK2GSK3BCDK9CCNT1CDK5
SCHEMBL23352055 0.79 CDK2 (0.33) CDK2GSK3BCDK9CCNT1CDK5
SCHEMBL15224899 0.77 KDM4E (0.42) CDK2CDK9CCNT1CDK5CDK5R1
SCHEMBL21481497 0.77 CDK2 (0.33) CDK2GSK3BCDK9CCNT1CDK5
SCHEMBL15224900 0.77 KDM4E (0.42) CDK2CDK9CCNT1CDK5CDK5R1
SCHEMBL30716366 0.77 DKK1 (0.37) HRH3HRH4CDK2GSK3BCDK9
SCHEMBL26973961 0.75 ALDH1A1 (0.40) CDK2CDK9CCNE1
SCHEMBL21481496 0.75 CDK2 (0.32) CDK2GSK3BCDK9CCNE1CDK7
SCHEMBL23381696 0.75 CDK2 (0.47) CDK2CDK9CCNT1CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019197549-A1 PYRAZOLO-TRIAZINE AND/OR PYRAZOLO-PYRIMIDINE DERIVATIVES AS SELECTIVE INHIBITOR OF CYCLIN DEPENDENT KINASE QURIENT CO., LTD. (KR) 2019-10-17 WO disclosed