SCHEMBL2149123

SCHEMBL2149123

Fc1ccc(F)c2c1CCOC2

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.33
SLC6A4 P31645 2/20 0.33
GRM2 Q14416 1/20 0.33
WNT3A P56704 1/20 0.32
TNKS2 Q9H2K2 1/20 0.32
ANO1 Q5XXA6 1/20 0.31
UGCG Q16739 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL33526079 0.86 IL1RN (0.33) GRM2WNT3ATNKS2
SCHEMBL2149255 0.74 DRD2 (0.44)
SCHEMBL1550867 0.74 HTR2A (0.34) HTR2AGRM2WNT3ATNKS2
SCHEMBL33526989 0.73 KDM1A (0.32) GRM2WNT3ATNKS2
SCHEMBL31518138 0.70 ABCC9 (0.36)
SCHEMBL23976544 0.69 SRD5A1 (0.39) HTR2A
SCHEMBL30060662 0.69 SRD5A1 (0.39) HTR2A
SCHEMBL30062825 0.69 DRD2 (0.33)
SCHEMBL23976551 0.69 DRD2 (0.33)
SCHEMBL30977517 0.68 HTR2A (0.39) HTR2ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2342182-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. Lundbeck A/S (DK) 2011-07-13 EP disclosed
WO-2010028655-A1 ISOQUINOLINONE DERIVATIVES AS NK3 ANTAGONISTS H. LUNDBECK A/S (DK) 2010-03-18 WO disclosed