SCHEMBL21494949

SCHEMBL21494949

NCCc1ccc(F)c(C2CC2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.57
BACE1 P56817 1/20 0.57
TAAR1 Q96RJ0 10/20 0.45
SLC6A2 P23975 3/20 0.42
SLC6A3 Q01959 3/20 0.42
SLC6A4 P31645 1/20 0.42
KDM4E B2RXH2 3/20 0.42
ATM Q13315 1/20 0.42
MAPK1 P28482 3/20 0.41
ADRA2A P08913 2/20 0.41
MAPT P10636 2/20 0.41
DRD2 P14416 2/20 0.41
DRD1 P21728 2/20 0.41
DRD4 P21917 2/20 0.41
DRD5 P21918 2/20 0.41
DRD3 P35462 2/20 0.41
RECQL P46063 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
PNMT P11086 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL62964 0.87 NUDT1 (0.42) NUDT1BACE1TAAR1SLC6A2SLC6A3
Hydrochloric Acid SCHEMBL52192 0.85 NUDT1 (0.41) NUDT1BACE1SLC6A2SLC6A3SLC6A4
SCHEMBL26032266 0.80 NUDT1 (0.47) NUDT1BACE1SLC6A2SLC6A3SLC6A4
SCHEMBL31734454 0.79 SOS1 (0.38) NUDT1BACE1SLC6A2SLC6A3SLC6A4
SCHEMBL18295013 0.79 SOS1 (0.40) NUDT1BACE1TAAR1SLC6A2SLC6A3
SCHEMBL16344820 0.79 CYP4F2 (0.45) NUDT1BACE1SLC6A2SLC6A3SLC6A4
SCHEMBL15614975 0.78 NUDT1 (0.53) NUDT1BACE1TAAR1SLC6A2SLC6A3
SCHEMBL12329238 0.77 NUDT1 (0.45) NUDT1BACE1SLC6A2SLC6A3SLC6A4
SCHEMBL21494904 0.76 SOS1 (0.36) NUDT1BACE1SLC6A2SLC6A3SLC6A4
SCHEMBL17186198 0.76 NUDT1 (0.51) NUDT1BACE1TAAR1SLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3781565-A1 2-METHYL-AZA-QUINAZOLINES Bayer Pharma Aktiengesellschaft (DE) 2021-02-24 EP disclosed
WO-2019201848-A1 2-METHYL-AZA-QUINAZOLINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2019-10-24 WO disclosed
CN-101379022-B Benzamide and heteroarene derivatives HOFFMANN LA ROCHE 2013-05-01 CN disclosed
CN-101379022-A Benzamide and heteroarene derivatives HOFFMANN LA ROCHE (CH) 2009-03-04 CN disclosed