SCHEMBL21494904

SCHEMBL21494904

O=CCc1ccc(F)c(C2CC2)c1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 1/20 0.36
NUDT1 P36639 1/20 0.34
BACE1 P56817 1/20 0.34
SCN9A Q15858 1/20 0.32
HCRTR2 O43614 1/20 0.32
HTR6 P50406 1/20 0.32
OPRL1 P41146 4/20 0.31
SLC6A2 P23975 2/20 0.31
SLC6A4 P31645 2/20 0.31
SLC6A3 Q01959 2/20 0.31
HTR1A P08908 1/20 0.31
PANK3 Q9H999 1/20 0.30
AKR1A1 P14550 1/20 0.30
AKR1B1 P15121 1/20 0.30
KDM1A O60341 2/20 0.30
KDM1B Q8NB78 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17675300 0.86 PANK3 (0.40) HTR6OPRL1PANK3
SCHEMBL62964 0.78 NUDT1 (0.42) SOS1NUDT1BACE1SLC6A2SLC6A4
SCHEMBL18295013 0.78 SOS1 (0.40) SOS1NUDT1BACE1HCRTR2HTR6
SCHEMBL31734454 0.78 SOS1 (0.38) SOS1NUDT1BACE1SCN9AHCRTR2
SCHEMBL16344820 0.78 CYP4F2 (0.45) SOS1NUDT1BACE1SCN9AHTR6
Hydrochloric Acid SCHEMBL52192 0.76 NUDT1 (0.41) SOS1NUDT1BACE1SLC6A2SLC6A4
SCHEMBL21494949 0.76 NUDT1 (0.57) NUDT1BACE1SLC6A2SLC6A4SLC6A3
SCHEMBL25388637 0.75 NOTUM (0.43) OPRL1
SCHEMBL21495043 0.75 ALDH1A1 (0.47)
SCHEMBL896163 0.74 HTT (0.42) KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3781565-A1 2-METHYL-AZA-QUINAZOLINES Bayer Pharma Aktiengesellschaft (DE) 2021-02-24 EP disclosed
WO-2019201848-A1 2-METHYL-AZA-QUINAZOLINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2019-10-24 WO disclosed