SCHEMBL21495098

SCHEMBL21495098

CC(=O)Nc1nc(-c2cccc(C)n2)cs1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.59
KDM4E B2RXH2 3/20 0.59
HSD17B10 Q99714 3/20 0.59
MAPK1 P28482 2/20 0.59
ABL1 P00519 7/20 0.59
RAB9A P51151 5/20 0.57
MAPT P10636 3/20 0.57
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
NFKB1 P19838 2/20 0.57
NFKB2 Q00653 2/20 0.57
RELA Q04206 2/20 0.57
STAT1 P42224 1/20 0.57
ALDH1A1 P00352 3/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
HTT P42858 2/20 0.55
HPGD P15428 1/20 0.55
LMNA P02545 1/20 0.55
POLB P06746 1/20 0.55
TYR P14679 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26122412 0.90 MRE11 (0.53) NPC1KDM4EHSD17B10MAPK1ABL1
SCHEMBL30313761 0.84 NPC1 (0.58) NPC1KDM4EHSD17B10MAPK1ABL1
SCHEMBL21484645 0.80 ABL1 (0.57) NPC1KDM4EMAPK1ABL1RAB9A
SCHEMBL26122183 0.80 CCR1 (0.55) NPC1KDM4ERAB9AMAPTMEN1
SCHEMBL17716927 0.79 ALDH1A1 (0.75) NPC1KDM4EHSD17B10MAPK1RAB9A
SCHEMBL30772147 0.77 ABL1 (0.76) NPC1KDM4EHSD17B10MAPK1ABL1
SCHEMBL2020280 0.77 ABL1 (0.73) NPC1KDM4EHSD17B10MAPK1ABL1
SCHEMBL22305595 0.76 MAPK1 (0.51) NPC1KDM4EMAPK1RAB9AMAPT
SCHEMBL28200307 0.76 ABL1 (0.76) NPC1KDM4EHSD17B10MAPK1ABL1
SCHEMBL19994395 0.76 MAPT (0.66) NPC1KDM4EHSD17B10RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019201867-A1 SUBSTITUTED PROPANAMIDES AS INHIBITORS OF NUCLEASES MASARYKOVA UNIVERZITA (CZ) 2019-10-24 WO disclosed