SCHEMBL21501014

SCHEMBL21501014

COC(=O)[C@H](Cc1ccc(F)cc1)N1C(=O)c2ccccc2C1=O

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.56
GAA P10253 2/20 0.56
HSD11B1 P28845 1/20 0.55
POLB P06746 3/20 0.54
KMT2A Q03164 4/20 0.54
L3MBTL1 Q9Y468 1/20 0.53
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
MAPT P10636 1/20 0.47
MEN1 O00255 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
PKM P14618 1/20 0.47
HTT P42858 1/20 0.46
CA12 O43570 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21501052 0.89 HSD11B1 (0.67) ALDH1A1GAAHSD11B1POLBKMT2A
SCHEMBL19597541 0.89 ALDH1A1 (0.70) ALDH1A1GAAHSD11B1POLBKMT2A
SCHEMBL19597540 0.89 ALDH1A1 (0.70) ALDH1A1GAAHSD11B1POLBKMT2A
SCHEMBL21501050 0.87 ALDH1A1 (0.56) ALDH1A1GAAHSD11B1POLBKMT2A
SCHEMBL1597751 0.87 ALDH1A1 (0.57) ALDH1A1GAAHSD11B1POLBKMT2A
SCHEMBL21501019 0.87 ALDH1A1 (0.56) ALDH1A1GAAHSD11B1POLBKMT2A
SCHEMBL23201840 0.86 MAPT (0.58) ALDH1A1GAAHSD11B1POLBKMT2A
SCHEMBL21501021 0.86 MAPT (0.58) ALDH1A1GAAHSD11B1POLBKMT2A
SCHEMBL6635286 0.83 ALDH1A1 (0.80) ALDH1A1GAAPOLBKMT2AL3MBTL1
SCHEMBL21914164 0.83 ALDH1A1 (0.80) ALDH1A1GAAPOLBKMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019204477-A1 PD(II)-CATALYZED ENANTIOSELECTIVE C-H ARYLATION OF FREE CARBOXYLIC ACIDS THE SCRIPPS RESEARCH INSTITUTE (US) 2019-10-24 WO disclosed