SCHEMBL21501554

SCHEMBL21501554

CN(CCNc1nc(Cl)ncc1Br)C(=O)C1CCC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 12/20 0.55
IKBKE Q14164 3/20 0.44
AURKB Q96GD4 3/20 0.44
CDK2 P24941 2/20 0.44
PDPK1 O15530 2/20 0.40
STK17A Q9UEE5 3/20 0.39
MARK4 Q96L34 2/20 0.39
MARK3 P27448 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
STK17B O94768 1/20 0.34
POLB P06746 1/20 0.34
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
RIPK1 Q13546 1/20 0.33
VHL P40337 1/20 0.32
ELOC Q15369 1/20 0.32
ELOB Q15370 1/20 0.32
HIF1A Q16665 1/20 0.32
IGF1R P08069 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17162049 0.94 TBK1 (0.63) TBK1IKBKEAURKBCDK2PDPK1
SCHEMBL29666237 0.94 TBK1 (0.63) TBK1IKBKEAURKBCDK2PDPK1
SCHEMBL23331357 0.89 TBK1 (0.58) TBK1IKBKEAURKBCDK2PDPK1
SCHEMBL22818571 0.82 TBK1 (0.51) TBK1IKBKEAURKBCDK2PDPK1
SCHEMBL22882524 0.80 TBK1 (0.65) TBK1IKBKEAURKBCDK2PDPK1
SCHEMBL22818563 0.80 TBK1 (0.49) TBK1IKBKEAURKBCDK2PDPK1
SCHEMBL1284852 0.78 TBK1 (0.61) TBK1IKBKEAURKBCDK2PDPK1
SCHEMBL23330925 0.77 STK17A (0.50) TBK1IKBKEAURKBCDK2STK17A
SCHEMBL21162388 0.77 TBK1 (0.90) TBK1IKBKEAURKBCDK2PDPK1
SCHEMBL3448808 0.76 MEN1 (0.47) STK17AMEN1KMT2ASTK17B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019201123-A1 MULTIFUNCTIONAL COMPOUND, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF IN PHARMACEUTICALS 四川科伦博泰生物医药股份有限公司 2019-10-24 WO disclosed