SCHEMBL2152525

SCHEMBL2152525

C=CCNC(=O)c1nc(C(=O)NCC=C)nc(C(=O)NCC=C)n1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.53
RAB9A P51151 2/20 0.48
HPGD P15428 10/20 0.47
ALDH1A1 P00352 3/20 0.47
TP53 P04637 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CYP1A2 P05177 4/20 0.46
LMNA P02545 2/20 0.46
TSHR P16473 1/20 0.45
MAPT P10636 1/20 0.45
PKM P14618 2/20 0.45
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
CYP3A4 P08684 3/20 0.44
CYP2C19 P33261 3/20 0.44
CYP2C9 P11712 2/20 0.44
POLB P06746 1/20 0.43
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16015011 0.78 SMN1; SMN2 (0.54) SMN1; SMN2RAB9AHPGDALDH1A1TP53
SCHEMBL2385213 0.73 HPGD (0.76) SMN1; SMN2RAB9AHPGDALDH1A1CYP1A2
SCHEMBL7112031 0.73 RAB9A (0.75) SMN1; SMN2RAB9AHPGDALDH1A1CYP1A2
SCHEMBL23309638 0.71 RAB9A (0.60) SMN1; SMN2RAB9AHPGDALDH1A1TP53
SCHEMBL29510 0.70
SCHEMBL627164 0.70 SMN1; SMN2 (0.47) SMN1; SMN2RAB9AHPGDALDH1A1TP53
SCHEMBL2152533 0.70 HPGD (0.49) SMN1; SMN2RAB9AHPGDALDH1A1TP53
SCHEMBL9426481 0.70 PKM (0.63) SMN1; SMN2RAB9AHPGDALDH1A1CYP1A2
SCHEMBL28489211 0.70 SMN1; SMN2 (1.00) SMN1; SMN2RAB9AHPGDALDH1A1L3MBTL1
SCHEMBL11419815 0.70 SMN1; SMN2 (0.50) SMN1; SMN2RAB9AHPGDALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 49 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2052041-B1 MULTI-LAYER COMPOSITES FORMED FROM COMPOSITIONS HAVING IMPROVED ADHESION PPG IND OHIO INC (US) 2019-10-09 EP disclosed
EP-1042402-B2 CURABLE FILM-FORMING COMPOSITIONS PPG IND OHIO INC (US) 2013-10-30 EP disclosed
EP-2397525-A2 Coating comprising terpene PPG Industries Ohio, Inc. (US) 2011-12-21 EP disclosed
US-8029894-B2 Multi-layer composites formed from compositions having improved adhesion PPG INDUSTRIES OHIO, INC. (US) 2011-10-04 US disclosed
US-20110165418-A1 MULTI-LAYER COMPOSITES FORMED FROM COMPOSITIONS HAVING IMPROVED ADHESION PPG INDUSTRIES OHIO, INC. 2011-07-07 US disclosed
EP-1417273-B1 COATING COMPOSITIONS HAVING IMPROVED ADHESION, COATED SUBSTRATES AND METHODS RELATED THERETO PPG IND OHIO INC (US) 2010-09-15 EP disclosed
US-7776959-B2 Coatings comprising terpene PPG INDUSTRIES OHIO, INC. (US) 2010-08-17 US disclosed
US-7737223-B2 Coating compositions containing amine-hydroxy functional polymer and/or amine-carbamate functional polymer PPG INDUSTRIES OHIO, INC. (US) 2010-06-15 US disclosed
EP-2092025-A2 COATINGS COMPRISING TERPENE PPG Industries Ohio, Inc. (US) 2009-08-26 EP disclosed
EP-2052041-A2 MULTI-LAYER COMPOSITES FORMED FROM COMPOSITIONS HAVING IMPROVED ADHESION PPG Industries Ohio, Inc. (US) 2009-04-29 EP disclosed
EP-1204701-A1 CURED COATINGS HAVING IMPROVED SCRATCH RESISTANCE, COATED SUBSTRATES AND METHODS RELATED THERETO PPG Industries Ohio, Inc. (US) 2002-05-15 EP disclosed
EP-1204709-A1 COATING COMPOSITIONS HAVING IMPROVED SCRATCH RESISTANCE, COATED SUBSTRATES AND METHODS RELATED THERETO PPG Industries Ohio, Inc. (US) 2002-05-15 EP disclosed
US-6387519-B1 CURED COMPOSITION COMPRISING PLURALITY OF PARTICLES, WHEREIN CONCENTRATION OF PARTICLES IN SURFACE REGION IS GREATER THAN THAT IN BULK REGION, AND COMPOSITION IS CURED BY EXPOSURE TO IONIZING RADIATION OR ACTINIC RADIATION WITH THERMAL ENERGY PPG INDUSTRIES OHIO, INC. 2002-05-14 US disclosed
WO-2002010298-A1 COATING COMPOSITIONS COMPRISING SILYL BLOCKED COMPONENTS, COATINGS, COATED SUBSTRATES AND METHODS RELATED THERETO PPG INDUSTRIES OHIO, INC. (US) 2002-02-07 WO disclosed
WO-2001009260-A1 COATING COMPOSITIONS HAVING IMPROVED SCRATCH RESISTANCE, COATED SUBSTRATES AND METHODS RELATED THERETO PPG INDUSTRIES OHIO, INC. (US) 2001-02-08 WO disclosed
WO-2001009259-A1 COATING COMPOSITIONS HAVING IMPROVED SCRATCH RESISTANCE, COATED SUBSTRATES AND METHODS RELATED THERETO PPG INDUSTRIES OHIO, INC. (US) 2001-02-08 WO disclosed
WO-2001009231-A1 CURED COATINGS HAVING IMPROVED SCRATCH RESISTANCE, COATED SUBSTRATES AND METHODS RELATED THERETO PPG INDUSTRIES OHIO, INC. (US) 2001-02-08 WO disclosed
EP-1042402-A1 CURABLE FILM-FORMING COMPOSITIONS PPG Industries Ohio, Inc. (US) 2000-10-11 EP disclosed
US-5965670-A COMPRISES ACRYLIC POLYOLS, AMINOPLAST AND CARBAMOYL TRIAZINES PPG INDUSTRIES OHIO, INC. (US) 1999-10-12 US disclosed
WO-1999033915-A1 CURABLE FILM-FORMING COMPOSITIONS PPG INDUSTRIES OHIO, INC. (US) 1999-07-08 WO disclosed