SCHEMBL2152808

SCHEMBL2152808

O=[N+]([O-])c1cc([As](=O)(O)O)ccc1F

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 7/20 0.67
MAPT P10636 4/20 0.67
KDM4E B2RXH2 2/20 0.67
L3MBTL1 Q9Y468 2/20 0.67
CYP2C19 P33261 2/20 0.67
USP2 O75604 1/20 0.67
PHPT1 Q9NRX4 1/20 0.67
ALDH1A1 P00352 6/20 0.55
HIF1A Q16665 1/20 0.55
MEN1 O00255 4/20 0.52
KMT2A Q03164 4/20 0.52
VCAM1 P19320 1/20 0.51
TDP1 Q9NUW8 2/20 0.51
POLB P06746 1/20 0.51
HTT P42858 3/20 0.44
CA1 P00915 1/20 0.44
MMP2 P08253 1/20 0.44
CA14 Q9ULX7 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Roxarsone SCHEMBL29485898 0.80 MAPT (1.00) LMNAMAPTKDM4EL3MBTL1CYP2C19
Roxarsone SCHEMBL28105454 0.80 MAPT (1.00) LMNAMAPTKDM4EL3MBTL1CYP2C19
Roxarsone SCHEMBL158026 0.80 MAPT (1.00) LMNAMAPTKDM4EL3MBTL1CYP2C19
Roxarsone SCHEMBL27915909 0.79 MAPT (0.96) LMNAMAPTKDM4EL3MBTL1CYP2C19
Roxarsone SCHEMBL20636782 0.79 MAPT (0.96) LMNAMAPTKDM4EL3MBTL1CYP2C19
SCHEMBL30986730 0.74 CYP2C19 (0.50) LMNAMAPTKDM4EL3MBTL1CYP2C19
SCHEMBL29385509 0.73 ALDH1A1 (0.62) LMNAMAPTALDH1A1HIF1AMEN1
SCHEMBL1187891 0.73 ALDH1A1 (0.62) LMNAMAPTALDH1A1HIF1AMEN1
SCHEMBL12625747 0.73 ALDH1A1 (0.56) LMNAMAPTALDH1A1HIF1AMEN1
SCHEMBL1858467 0.73 ALDH1A1 (0.56) LMNAMAPTALDH1A1HIF1AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1228076-B1 A SUBSTANTIALLY CELL MEMBRANE IMPERMEABLE COMPOUND AND USE THEREOF NEWSOUTH INNOVATIONS PTY LTD (AU) 2011-07-06 EP disclosed