Loratadine

Loratadine

SCHEMBL21529220

CCOC(=O)N1CCC(=C2c3ccc(Cl)cc3CCc3cccnc32)CC1.[Mn]

nearest known ligand 0.98

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HRH1

The experimentally established mechanism targets of Loratadine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 known ✓ P35367 8/20 0.98
SLC6A15 Q9H2J7 15/20 0.98
MEN1 O00255 1/20 0.98
NPC1 O15118 1/20 0.98
CACNA1F O60840 1/20 0.98
NR1I2 O75469 1/20 0.98
GMNN O75496 1/20 0.98
USP2 O75604 1/20 0.98
ABCB11 O95342 1/20 0.98
LMNA P02545 1/20 0.98
TP53 P04637 1/20 0.98
CHRM2 P08172 1/20 0.98
ABCB1 P08183 1/20 0.98
CYP3A4 P08684 1/20 0.98
ADORA3 P0DMS8 1/20 0.98
CYP2C8 P10632 1/20 0.98
CYP2D6 P10635 1/20 0.98
MAPT P10636 1/20 0.98
CYP2C9 P11712 1/20 0.98
ADRB3 P13945 1/20 0.98

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Loratadine SCHEMBL29380223 0.99 SLC6A15 (1.00) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL3862958 0.99 SLC6A15 (1.00) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL29441811 0.99 SLC6A15 (1.00) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL4596 0.99 SLC6A15 (1.00) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL2166756 0.98 SLC6A15 (0.98) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL21529200 0.98 SLC6A15 (0.98) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL21529218 0.98 SLC6A15 (0.98) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL28800563 0.98 SLC6A15 (0.98) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL28594875 0.98 SLC6A15 (0.98) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL28123874 0.98 SLC6A15 (0.98) SLC6A15HRH1MEN1NPC1CACNA1F

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11357802-B2 Oral delivery compositions for improved gut barrier protection and immunity in mammals VETS PLUS, INC. (US) 2022-06-14 US disclosed
US-20190336546-A1 ORAL DELIVERY COMPOSITIONS FOR IMPROVED GUT BARRIER PROTECTION AND IMMUNITY IN MAMMALS VETS PLUS, INC. (US) 2019-11-07 US disclosed