Loratadine

Loratadine

SCHEMBL4596

CCOC(=O)N1CCC(=C2c3ccc(Cl)cc3CCc3cccnc32)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HRH1

The experimentally established mechanism targets of Loratadine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 known ✓ P35367 8/20 1.00
SLC6A15 Q9H2J7 15/20 1.00
MEN1 O00255 1/20 1.00
NPC1 O15118 1/20 1.00
CACNA1F O60840 1/20 1.00
NR1I2 O75469 1/20 1.00
GMNN O75496 1/20 1.00
USP2 O75604 1/20 1.00
ABCB11 O95342 1/20 1.00
LMNA P02545 1/20 1.00
TP53 P04637 1/20 1.00
CHRM2 P08172 1/20 1.00
ABCB1 P08183 1/20 1.00
CYP3A4 P08684 1/20 1.00
ADORA3 P0DMS8 1/20 1.00
CYP2C8 P10632 1/20 1.00
CYP2D6 P10635 1/20 1.00
MAPT P10636 1/20 1.00
CYP2C9 P11712 1/20 1.00
ADRB3 P13945 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Loratadine SCHEMBL29380223 1.00 SLC6A15 (1.00) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL29441811 1.00 SLC6A15 (1.00) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL3862958 1.00 SLC6A15 (1.00) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL2166756 0.99 SLC6A15 (0.98) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL21529220 0.99 SLC6A15 (0.98) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL28800563 0.99 SLC6A15 (0.98) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL21529200 0.99 SLC6A15 (0.98) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL21529218 0.99 SLC6A15 (0.98) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL28594875 0.99 SLC6A15 (0.98) SLC6A15HRH1MEN1NPC1CACNA1F
Loratadine SCHEMBL27891063 0.99 SLC6A15 (0.98) SLC6A15HRH1MEN1NPC1CACNA1F

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 46995 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-121265587-B Use of oligomycin A for the preparation of a medicament for the competitive inhibition of EphB3 for reversing the resistance of Loratinib AFFILIATED HOSPITAL OF NANTONG UNIVERSITY (CN) 2026-05-26 CN claimed
WO-2026104580-A1 PHARMACEUTICAL COMPOSITIONS USING NON-ANIMAL ORIGIN MATRIX FORMERS AND METHODS OF MAKING THEREOF CATALENT U.K. SWINDON ZYDIS LIMITED (GB) 2026-05-21 WO claimed
WO-2026100654-A1 NUCLEIC ACID INTRODUCTION AID, NUCLEIC ACID INTRODUCTION AGENT, AND NUCLEIC ACID INTRODUCTION METHOD 株式会社インファーマシア 2026-05-15 WO claimed
US-20260131006-A1 PHARMACEUTICAL COMPOSITIONS USING NON-ANIMAL ORIGIN MATRIX FORMERS AND METHODS OF MAKING THEREOF CATALENT U.K. SWINDON ZYDIS LIMITED (GB) 2026-05-14 US claimed
EP-4736841-A1 A MUCOADHESIVE LAYER FOR BUCCAL ADMINISTRATION OF AN ACTIVE PHARMACEUTICAL INGREDIENT IQ medical GmbH (DE) 2026-05-06 EP claimed
EP-4734952-A1 ORAL TABLET WITH IMPROVED UNIFORMITY OF CONTENT OF ACTIVES Fertin Pharma A/S (DK) 2026-05-06 EP claimed
US-20260115192-A1 PHARMACEUTICAL COMPOSITIONS SHENZHEN PHARMACIN CO LTD (CN) 2026-04-30 US claimed
US-20260115161-A1 2-HYDROXY-OCTADECENE-9-CIS-OATE FOR USE IN THE TREATMENT OF ONCOLOGICAL PATHOLOGIES AND NEUROPATHIC PAIN LAMINAR PHARMACEUTICALS S A (ES) 2026-04-30 US claimed
EP-4724049-A1 MODIFIED RELEASE FILL COMPOSITIONS FOR DOSAGE FORMS AND METHODS OF PREPARATION AND USE THEREOF Catalent Ontario Limited (CA) 2026-04-15 EP claimed
US-20260097039-A1 METHODS FOR TREATING A FATTY LIVER DISEASE MADRIGAL PHARMACEUTICALS INC (US) 2026-04-09 US claimed
EP-0050336-A1 Panel file used for storage of mainly rectangular relatively thin sheets, in particular microfiche Thomsen, Preben West (DK) 1982-04-28 EP claimed
EP-0046588-A1 Method of and circuit arrangement for supplying current to a two-wire telecommunications line International Standard Electric Corporation (US) 1982-03-03 EP claimed
EP-0044885-A1 Method and apparatus for determining at least one geometrical characteristic of the rail heads of a railway track SPENO INTERNATIONAL S.A. (CH) 1982-02-03 EP claimed
EP-0042544-A2 Novel antihistamines, process for their preparation and pharmaceutical compositions containing them SCHERING CORPORATION (US) 1981-12-30 EP claimed
US-4282233-A NO SEDATIVE EFFECT SCHERING CORPORATION (US) 1981-08-04 US claimed
EP-0010018-A1 Method and apparatus for producing a small quadrangular flat bag and for filling this bag with a solid or liquid substance of a predetermined quantity SOCIETE DES ETABLISSEMENTS THIMON (FR) 1980-04-16 EP claimed
EP-0007343-A1 METHOD AND APPARATUS FOR REGENERATING FILTERS ENVIRONMENTAL INDUSTRIAL PRODUCTS, INC. (US) 1980-02-06 EP claimed
WO-1979000655-A1 BAND OF BAGS,PROCESS AND DEVICE FOR PRODUCING SUCH SCHERZ W (DE) 1979-09-06 WO claimed
EP-0003197-A1 Grinding machine for very hard workpieces SOCIETE EUROPEENNE DES PRODUITS REFRACTAIRES (FR) 1979-07-25 EP claimed
WO-1979000086-A1 METHOD AND APPARATUS FOR REGENERATING FILTERS ENVIRONMENTAL IND PROD (US) 1979-02-22 WO claimed