SCHEMBL21538245

SCHEMBL21538245

COc1ccc(OC)c(CN2CCN(C)CC2)c1

nearest known ligand 0.71

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.67
TSHR P16473 1/20 0.67
TP53 P04637 1/20 0.61
NPC1 O15118 1/20 0.60
ALDH1A1 P00352 1/20 0.57
GAA P10253 1/20 0.56
RECQL P46063 1/20 0.56
MAPT P10636 1/20 0.55
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
HTR6 P50406 1/20 0.54
POLB P06746 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21650968 0.94 MEN1 (0.62) KDM4ETSHRTP53NPC1ALDH1A1
SCHEMBL21164680 0.88 KDM4E (0.64) KDM4ETSHRTP53NPC1ALDH1A1
SCHEMBL18182089 0.88 KDM4E (0.67) KDM4ETSHRTP53NPC1ALDH1A1
SCHEMBL9830022 0.87 KDM4E (0.68) KDM4ETSHRTP53NPC1ALDH1A1
SCHEMBL13256755 0.87 KDM4E (0.62) KDM4ETSHRTP53NPC1ALDH1A1
SCHEMBL20125154 0.84 MEN1 (0.57) KDM4ETSHRTP53ALDH1A1GAA
SCHEMBL18177824 0.84 KDM4E (0.62) KDM4ETSHRTP53NPC1ALDH1A1
SCHEMBL7300721 0.83 CYP1A2 (0.62) KDM4ETSHRTP53NPC1ALDH1A1
Hydrochloric Acid SCHEMBL7563307 0.82 NR1H2 (0.55) KDM4ETSHRGAAMEN1KMT2A
SCHEMBL15828705 0.81 ALDH1A1 (0.54) KDM4ETSHRALDH1A1GAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3561077-B1 METHODS FOR CELL-PROLIFERATION-RELATED DISORDERS SERVIER LAB (FR) 2022-12-21 EP disclosed
EP-3561077-A1 METHODS AND COMPOSITIONS FOR CELL-PROLIFERATION-RELATED DISORDERS Agios Pharmaceuticals, Inc. (US) 2019-10-30 EP disclosed