SCHEMBL21546549

SCHEMBL21546549

Bc1cc(Br)c2cc(Br)cc(Br)c2c1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.38
TSHR P16473 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRA2 P47869 1/20 0.33
GABRB2 P47870 1/20 0.33
AHR P35869 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30449010 0.83 TDP1 (0.50) CYP3A4TSHRTDP1GABRA1GABRB1
SCHEMBL4324429 0.83 TDP1 (0.50) CYP3A4TSHRTDP1GABRA1GABRB1
SCHEMBL21546553 0.72 CYP2A6 (0.33) CYP3A4TSHRTDP1
SCHEMBL10065756 0.70
SCHEMBL21546552 0.69 CYP3A4 (0.33) CYP3A4TSHRTDP1GABRA1GABRB1
SCHEMBL29010717 0.68 TDP1 (0.38) CYP3A4TSHRTDP1GABRA1GABRB1
SCHEMBL20356132 0.67 PARP1 (0.42) CYP3A4TSHRTDP1GABRA1GABRB1
SCHEMBL22601373 0.64 ALDH1A1 (0.41) CYP3A4TSHRTDP1AHR
SCHEMBL12165264 0.63 TSHR (0.35) TSHR
SCHEMBL27308331 0.63 TDP1 (0.43) CYP3A4TSHRTDP1GABRA1GABRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3564245-A1 NAPHTHOBISCHALCOGENADIAZOLE DERIVATIVE AND PRODUCTION METHOD THEREFOR Osaka University (JP) 2019-11-06 EP disclosed