SCHEMBL21546860

SCHEMBL21546860

Cc1ccccc1-c1ccc2c3ccc(-c4ccccc4C)cc3n(-c3cc(C#N)c(-c4cccc(C#N)c4)cc3-n3c4cc(-c5ccccc5C)ccc4c4ccc(-c5ccccc5C)cc43)c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.42
ADRA2C P18825 1/20 0.38
BRD4 O60885 1/20 0.37
GABRA1 P14867 2/20 0.35
GABRG2 P18507 2/20 0.35
GABRB3 P28472 2/20 0.35
GABRA2 P47869 2/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
HTR1A P08908 1/20 0.34
HTR7 P34969 1/20 0.34
ALDH1A3 P47895 1/20 0.34
MEN1 O00255 2/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C19 P33261 2/20 0.34
KMT2A Q03164 2/20 0.34
CLK4 Q9HAZ1 2/20 0.34
CYP11B1 P15538 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21546858 0.97 AR (0.40) ARADRA2CBRD4GABRA1GABRG2
SCHEMBL21546957 0.92 AR (0.41) ARADRA2CBRD4GABRA1GABRG2
SCHEMBL21546672 0.91 AR (0.42) ARADRA2CBRD4GABRA1GABRG2
SCHEMBL21546859 0.90 AR (0.40) ARADRA2CBRD4GABRA1GABRG2
SCHEMBL21546955 0.90 AR (0.40) ARADRA2CBRD4GABRA1GABRG2
SCHEMBL22760959 0.90 TRPA1 (0.41) ADRA2CGABRA1GABRG2GABRB3GABRA2
SCHEMBL22760967 0.90 ALDH1A3 (0.39) ARADRA2CBRD4ALDH1A3ALDH1A1
SCHEMBL21546689 0.89 ALDH1A3 (0.42) ADRA2CGABRA1GABRG2GABRB3GABRA5
SCHEMBL21546662 0.88 AR (0.41) ARBRD4ALDH1A3ALDH1A1CYP1A2
SCHEMBL22760961 0.87 ALDH1A3 (0.39) ADRA2CALDH1A3MEN1ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3478793-B1 ORGANIC MOLECULES, IN PARTICULAR FOR USE IN OPTOELECTRONIC DEVICES CYNORA GMBH (DE) 2019-11-06 EP disclosed