SCHEMBL21550141

SCHEMBL21550141

CCS(=O)(=O)Cc1ccc(C(=O)c2cccc(Cl)c2Cl)c(-c2cn(C)c(=O)cc2CNC(=O)OC(C)(C)C)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 4/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35
DRD2 P14416 4/20 0.34
POLB P06746 1/20 0.34
MAPK1 P28482 1/20 0.34
ATM Q13315 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
CYP2C9 P11712 1/20 0.33
KCNA5 P22460 1/20 0.33
HTT P42858 1/20 0.32
KIF18A Q8NI77 1/20 0.32
DRD3 P35462 1/20 0.32
LMNA P02545 1/20 0.32
HPGD P15428 1/20 0.32
ALDH2 P05091 1/20 0.32
BRD9 Q9H8M2 1/20 0.32
BAZ2B Q9UIF8 1/20 0.32
BAZ2A Q9UIF9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21564924 0.94 HDAC10 (0.36) POLBMAPK1ATMHDAC10HDAC6
SCHEMBL21550125 0.90 ALDH1A1 (0.36) PKMCYP1A2CYP2C19POLBMAPK1
SCHEMBL21550252 0.90 ALDH1A1 (0.34) PKMDRD2HDAC10HDAC6KCNA5
SCHEMBL20157852 0.89 BRD4 (0.36) PKMCYP2C19HDAC10HDAC6
SCHEMBL21564753 0.88 POLB (0.38) PKMCYP1A2CYP2C19DRD2POLB
SCHEMBL20157351 0.88 HDAC10 (0.36) CYP2C19DRD2HDAC10HDAC6CYP2C9
SCHEMBL21550059 0.87 NAMPT (0.33) POLBMAPK1ATMHDAC10HDAC6
SCHEMBL20157909 0.87 BRD4 (0.34) CYP2C19HDAC10HDAC6CYP2C9HTT
SCHEMBL21362637 0.86 BRD4 (0.33) HDAC10HDAC6BAZ2BBAZ2A
SCHEMBL20158039 0.85 BRD4 (0.34) HDAC10HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019214399-A1 BENZO- SEVEN-MEMBERED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATION THEREOF 罗欣药业(上海)有限公司 (CN) 2019-11-14 WO disclosed
WO-2019214399-A1 BENZO- SEVEN-MEMBERED HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATION THEREOF 罗欣药业(上海)有限公司 (CN) 2019-11-14 WO disclosed