SCHEMBL21362637

SCHEMBL21362637

CCS(=O)(=O)Cc1ccc(C(=O)c2cc(OC)c(C)cc2Cl)c(-c2cn(C)c(=O)cc2CNC(=O)OC(C)(C)C)c1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.33
BAZ2B Q9UIF8 1/20 0.31
BAZ2A Q9UIF9 1/20 0.31
PDE10A Q9Y233 1/20 0.30
SUV39H2 Q9H5I1 4/20 0.30
HDAC10 Q969S8 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
RAF1 P04049 1/20 0.30
BRAF P15056 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
TSHR P16473 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20158039 0.92 BRD4 (0.34) BRD4SUV39H2HDAC10HDAC6
SCHEMBL21550125 0.88 ALDH1A1 (0.36) BRD4BAZ2BBAZ2AHDAC10HDAC6
SCHEMBL21550252 0.88 ALDH1A1 (0.34) BRD4HDAC10HDAC6
SCHEMBL20157852 0.88 BRD4 (0.36) BRD4HDAC10HDAC6
SCHEMBL21564924 0.87 HDAC10 (0.36) BRD4BAZ2BBAZ2AHDAC10HDAC6
SCHEMBL21550141 0.86 PKM (0.36) BAZ2BBAZ2AHDAC10HDAC6
SCHEMBL21550059 0.85 NAMPT (0.33) BRD4HDAC10HDAC6
SCHEMBL21550010 0.84 BRD4 (0.36) BRD4HDAC10HDAC6RAF1BRAF
SCHEMBL20157351 0.84 HDAC10 (0.36) BRD4HDAC10HDAC6SMN1; SMN2
SCHEMBL20157909 0.84 BRD4 (0.34) BRD4HDAC10HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed