SCHEMBL21553676

SCHEMBL21553676

CNC(C)C(=O)NC(CC(N)=O)C(=O)N1CCCC1C(=O)NC(CN)C(N)=O

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
XIAP P98170 6/20 0.52
CAPN1 P07384 4/20 0.44
NMUR2 Q9GZQ4 2/20 0.42
NMUR1 Q9HB89 2/20 0.42
OPRM1 P35372 2/20 0.42
CTSB P07858 1/20 0.42
F2 P00734 1/20 0.40
F10 P00742 1/20 0.40
PLG P00747 1/20 0.40
PRSS1 P07477 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21553671 0.84 XIAP (0.42) XIAPCAPN1NMUR2NMUR1OPRM1
SCHEMBL29721089 0.77 CALCRL (0.46) XIAPOPRM1OPRD1OPRK1
SCHEMBL18098145 0.76 F2 (0.50) CAPN1NMUR2NMUR1OPRM1CTSB
SCHEMBL21310170 0.75 XIAP (0.45) XIAPNMUR2NMUR1F2F10
SCHEMBL30353032 0.75 F2 (0.42) NMUR2NMUR1OPRM1F2F10
SCHEMBL16508578 0.75 OPRM1 (0.49) XIAPNMUR2NMUR1OPRM1OPRK1
SCHEMBL16508495 0.75 OPRM1 (0.49) XIAPNMUR2NMUR1OPRM1OPRK1
SCHEMBL22623412 0.75 XIAP (0.70) XIAPOPRM1OPRD1OPRK1
SCHEMBL22942169 0.74 REN (0.42) XIAPCAPN1NMUR2NMUR1OPRM1
SCHEMBL31556402 0.74 CAPN1 (0.50) CAPN1NMUR2NMUR1OPRM1CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970390-B1 MACROCYCLIC INHIBITORS OF THE PD-1/PD-L1 AND CD80(B7-1)/PD-L1 PROTEIN/PROTEIN INTERACTIONS BRISTOL MYERS SQUIBB CO (US) 2019-11-06 EP disclosed