SCHEMBL21558093

SCHEMBL21558093

COc1cc(OCCN2CCN(C)CC2)c(N)cc1N

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.45
HTR1B P28222 1/20 0.44
POLB P06746 1/20 0.43
NOS3 P29474 3/20 0.43
NOS1 P29475 3/20 0.43
NOS2 P35228 3/20 0.43
SYK P43405 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
LTA4H P09960 2/20 0.41
EHMT2 Q96KQ7 1/20 0.41
EHMT1 Q9H9B1 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19175202 0.89 GAA (0.53) ABCB1POLBNOS3NOS1NOS2
SCHEMBL2204177 0.81 MEN1 (0.52) ABCB1MEN1KMT2ALTA4HKDM4E
SCHEMBL6313608 0.79 KDM4E (0.53) ABCB1HTR1BPOLBNOS3NOS1
SCHEMBL4042949 0.79 SLC29A1 (0.50) ABCB1HTR1BPOLBSYKMEN1
SCHEMBL15016438 0.79 HTR1B (0.47) ABCB1HTR1BNOS3NOS1NOS2
SCHEMBL6314286 0.79 SYK (0.56) ABCB1HTR1BPOLBSYKMEN1
SCHEMBL4088385 0.78 SYK (0.59) POLBSYK
SCHEMBL24179121 0.77 SIGMAR1 (0.48) POLBNOS3NOS1NOS2MEN1
SCHEMBL16803350 0.77 HTR1B (0.51) ABCB1HTR1BPOLBNOS3NOS1
SCHEMBL12409057 0.75 SMN1; SMN2 (0.57) ABCB1HTR1BPOLBSYKMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2844642-B1 COMPOUNDS FOR INHIBITING CELL PROLIFERATION IN EGFR-DRIVEN CANCERS ARIAD PHARMA INC (US) 2019-11-13 EP disclosed