SCHEMBL6314286

SCHEMBL6314286

COc1cc(N)cc(OC)c1OCCN1CCN(C)CC1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.56
POLB P06746 1/20 0.54
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
SLC29A1 Q99808 1/20 0.46
ALDH1A1 P00352 2/20 0.44
CYP2D6 P10635 2/20 0.44
CYP1A2 P05177 1/20 0.44
KDM4E B2RXH2 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ABCB1 P08183 1/20 0.43
TSHR P16473 1/20 0.43
HTR1B P28222 1/20 0.41
TERT O14746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4042949 0.91 SLC29A1 (0.50) SYKPOLBMEN1KMT2ASLC29A1
SCHEMBL6992013 0.89 POLB (0.68) SYKPOLBMEN1KMT2AALDH1A1
SCHEMBL12435658 0.85 SYK (0.77) SYKPOLBMEN1KMT2ACYP2D6
SCHEMBL6313608 0.82 KDM4E (0.53) POLBALDH1A1KDM4EABCB1HTR1B
SCHEMBL6313695 0.80 POLB (0.55) SYKPOLBMEN1KMT2ASLC29A1
SCHEMBL21558093 0.79 ABCB1 (0.45) SYKPOLBMEN1KMT2AALDH1A1
SCHEMBL2087346 0.78 CYP2D6 (0.71) SYKMEN1KMT2AALDH1A1CYP2D6
SCHEMBL19392831 0.77 SYK (0.61) SYKPOLBMEN1KMT2AALDH1A1
SCHEMBL4038948 0.77 CYP2D6 (0.65) SYKMEN1KMT2AALDH1A1CYP2D6
SCHEMBL2088116 0.77 SYK (0.65) SYKPOLBSLC29A1ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6939874-B2 Substituted pyrimidinyl derivatives and methods of use AMGEN INC. (US) 2005-09-06 US disclosed
US-20040063705-A1 Substituted pyrimidinyl derivatives and methods of use AMGEN INC. 2004-04-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040063705-A1 Substituted pyrimidinyl derivatives and methods of use DPYD, TYMP, TPMT SYK 928/4885POLB 944/4885MEN1 1164/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.