SCHEMBL21564573

SCHEMBL21564573

CNCCCc1cn(Cc2ccc(F)cc2)c(=O)c(N2CCN(C)CC2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.43
ALDH1A1 P00352 6/20 0.41
CYP3A4 P08684 6/20 0.41
HSD17B10 Q99714 5/20 0.41
GLA P06280 3/20 0.41
TSHR P16473 5/20 0.40
CYP1A2 P05177 3/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
USP2 O75604 5/20 0.39
MAPK1 P28482 2/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
HTR6 P50406 1/20 0.39
CASP1 P29466 4/20 0.38
CASP7 P55210 4/20 0.38
HIF1A Q16665 4/20 0.38
CYP2C19 P33261 1/20 0.38
FSCN1 Q16658 1/20 0.38
CYP2D6 P10635 1/20 0.38
BRD4 O60885 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21553124 0.87 HDAC6 (0.44) HDAC6ALDH1A1CYP3A4HSD17B10GLA
SCHEMBL23258582 0.87 HDAC6 (0.44) HDAC6ALDH1A1CYP3A4HSD17B10GLA
SCHEMBL21564887 0.87 SOS1 (0.36) HDAC6ALDH1A1FSCN1BRD4NPSR1
SCHEMBL21552877 0.84 KDM1A (0.45) HDAC6
SCHEMBL21553024 0.83 ALDH1A1 (0.45) HDAC6ALDH1A1CYP3A4HSD17B10GLA
SCHEMBL21552841 0.79 HDAC6 (0.48) HDAC6ALDH1A1CYP3A4HSD17B10GLA
SCHEMBL21553012 0.78 HDAC6 (0.43) HDAC6ALDH1A1CYP3A4HSD17B10GLA
SCHEMBL21564690 0.77 BRD4 (0.38) HDAC6ALDH1A1HSD17B10TSHRMAPK1
SCHEMBL21564541 0.76 CYP11B1 (0.41) HDAC6ALDH1A1FSCN1BRD4NPSR1
SCHEMBL23258706 0.76 ALDH1A1 (0.41) HDAC6ALDH1A1CYP3A4CYP2C19FSCN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019217972-A1 KDM1A INHIBITORS FOR THE TREATMENT OF DISEASE IMAGO BIOSCIENCES, INC. (US) 2019-11-14 WO disclosed