Phloretin

Phloretin

SCHEMBL2157151

COC1=C(O)C=CC(C=CC(=O)c2ccccc2O)C1.O=C(CCc1ccc(O)cc1)c1c(O)cc(O)cc1O

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC5A1 P13866 11/20 0.46
SLC5A2 P31639 8/20 0.46
CYP19A1 P11511 4/20 0.45
MAPT P10636 3/20 0.45
SLC28A3 Q9HAS3 3/20 0.45
HPGD P15428 3/20 0.45
HSD17B10 Q99714 3/20 0.45
NFKB1 P19838 2/20 0.45
NFKB2 Q00653 2/20 0.45
RELA Q04206 2/20 0.45
GAA P10253 2/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
KDM4E B2RXH2 2/20 0.45
CYP3A4 P08684 2/20 0.45
THRB P10828 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
SLC16A3 O15427 1/20 0.45
ALDH1A1 P00352 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3396798 0.83 MAOB (0.45) MAPTHPGDMEN1KMT2AKDM4E
SCHEMBL2023335 0.79 MEN1 (0.47) CYP19A1MAPTHPGDHSD17B10NFKB1
SCHEMBL2020902 0.78 SLC5A1 (0.43) SLC5A1SLC5A2CYP19A1MAPTHSD17B10
SCHEMBL2023203 0.73 AURKA (0.40) SLC5A1SLC5A2CYP19A1NFKB1NFKB2
SCHEMBL15313125 0.73 ALDH1A1 (0.45) KDM4EALDH1A1POLBACHE
SCHEMBL2024880 0.72 CAPN1 (0.44) MAPTMEN1KMT2AALDH1A1TDP1
Phloretin SCHEMBL21192491 0.70 SLC5A1 (0.87) SLC5A1SLC5A2CYP19A1MAPTSLC28A3
Phloretin SCHEMBL1260339 0.69 SLC5A1 (0.51) SLC5A1SLC5A2CYP19A1MAPTSLC28A3
SCHEMBL31527864 0.69 MAOB (0.45) MAPTHPGDMEN1KMT2AKDM4E
SCHEMBL27182973 0.69 MAOB (0.45) MAPTHPGDMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9198451-B2 Aroma composition to reduce or suppress undesirable bitter and astringent taste impressions of sweeteners SYMRISE AG (DE) 2015-12-01 US disclosed
EP-2340719-B1 Aroma composition comprising o-coumaric acid to reduce or suppress undesirable taste impressions of sweeteners SYMRISE AG (DE) 2014-02-19 EP disclosed
EP-2220945-B1 Aroma composition to reduce or suppress undesirable bitter and astringent taste impressions of sweeteners SYMRISE AG (DE) 2013-03-27 EP disclosed
EP-2340719-A1 Aroma composition comprising o-coumaric acid to reduce or suppress undesirable taste impressions of sweeteners Symrise AG (DE) 2011-07-06 EP disclosed
EP-2220945-A1 Aroma composition to reduce or suppress undesirable bitter and astringent taste impressions of sweeteners Symrise GmbH & Co. KG (DE) 2010-08-25 EP disclosed
US-20100151055-A1 Aroma Composition to Reduce or Suppress Undesirable Bitter and Astringent Taste Impressions of Sweeteners SYMRISE GMBH & CO. KG (DE) 2010-06-17 US disclosed