SCHEMBL21573641

SCHEMBL21573641

COc1cc(OC)c(-c2ccc(Cl)cc2F)cc1B1OC(C)(C)C(C)(C)O1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.45
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
TRPV4 Q9HBA0 1/20 0.32
LIPE Q05469 1/20 0.32
AMY1A P0DUB6 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.31
EZH2 Q15910 1/20 0.31
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31
CTSD P07339 1/20 0.31
BACE1 P56817 1/20 0.31
FGFR1 P11362 1/20 0.31
FLT1 P17948 1/20 0.31
EPHB2 P29323 1/20 0.31
FLT4 P35916 1/20 0.31
KDR P35968 1/20 0.31
LMNA P02545 1/20 0.30
GAA P10253 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20321544 0.83 EGFR (0.41) EGFR
SCHEMBL21573743 0.81 EGFR (0.42) EGFR
SCHEMBL21784550 0.78 EGFR (0.44) EGFRLMNAKMT2A
SCHEMBL16282205 0.78 EGFR (0.47) EGFRHSP90AA1HSP90AB1TRPV4LIPE
SCHEMBL5892464 0.78 EGFR (0.47) EGFRTRPV4LIPELMNAKMT2A
SCHEMBL20209464 0.78 HSP90AA1 (0.43) EGFRHSP90AA1HSP90AB1TRPV4AMY1A
SCHEMBL29695387 0.76 EGFR (0.52) EGFR
SCHEMBL2112318 0.76 EGFR (0.52) EGFR
SCHEMBL23772414 0.75 EGFR (0.45) EGFR
SCHEMBL2355702 0.75 LPL (0.40) EGFRLIPEROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3569603-A1 POLYCYCLIC COMPOUND, AND ORGANIC ELECTROLUMINESCENCE ELEMENT COMPRISING THE POLYCYCLIC COMPOUND Idemitsu Kosan Co., Ltd. (JP) 2019-11-20 EP disclosed