SCHEMBL21574952

SCHEMBL21574952

CC(=O)N[S+]([O-])c1cccc(CN(CCc2ccc(Br)cc2)C2CCN(c3nc(N)n[nH]3)CC2)c1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHIT1 Q13231 19/20 0.44
CHIA Q9BZP6 19/20 0.44
KCNH2 Q12809 13/20 0.44
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21575086 0.92 CHIT1 (0.47) CHIT1CHIAKCNH2
SCHEMBL21574951 0.90 CHIT1 (0.49) CHIT1CHIAKCNH2
SCHEMBL17838860 0.84 CHIT1 (0.45) CHIT1CHIAKCNH2
SCHEMBL17838853 0.83 CHIT1 (0.49) CHIT1CHIAKCNH2MEN1KMT2A
SCHEMBL17838868 0.81 CHIT1 (0.48) CHIT1CHIAKCNH2
SCHEMBL16826354 0.80 CHIA (0.59) CHIT1CHIAKCNH2MEN1KMT2A
SCHEMBL17838875 0.79 CHIT1 (0.50) CHIT1CHIAKCNH2
SCHEMBL17838869 0.78 CHIT1 (0.51) CHIT1CHIAKCNH2MEN1KMT2A
SCHEMBL17838895 0.78 CHIT1 (0.51) CHIT1CHIAKCNH2
SCHEMBL17838888 0.77 CHIT1 (0.51) CHIT1CHIAKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3233832-B1 SUBSTITUTED AMINO TRIAZOLES USEFUL AS ACIDIC MAMMALIAN CHITINASE INHIBITORS ONCOARENDI THERAPEUTICS SA (PL) 2019-11-20 EP disclosed