SCHEMBL21582154

SCHEMBL21582154

COc1cc([N+](=O)[O-])cc(Br)c1OC(C)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.44
HTT P42858 6/20 0.43
MAPT P10636 4/20 0.43
CRHBP P24387 1/20 0.43
CRHR2 Q13324 1/20 0.43
ALDH1A1 P00352 2/20 0.43
PKM P14618 3/20 0.43
KMT2A Q03164 1/20 0.41
TSHR P16473 1/20 0.41
APOBEC3A P31941 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
KRAS P01116 2/20 0.40
PTGS2 P35354 1/20 0.40
EPHX1 P07099 1/20 0.40
GAA P10253 1/20 0.40
VCP P55072 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
LMNA P02545 1/20 0.40
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17132381 0.84 HTT (0.50) ERN1HTTMAPTALDH1A1PKM
SCHEMBL29155725 0.83 ERN1 (0.44) ERN1HTTMAPTCRHBPCRHR2
SCHEMBL30318939 0.82 HTT (0.45) ERN1HTTMAPTALDH1A1PKM
SCHEMBL5565950 0.77 ALDH1A1 (0.50) ERN1HTTMAPTCRHBPCRHR2
SCHEMBL1437010 0.76 ERN1 (0.62) ERN1HTTMAPTALDH1A1PKM
SCHEMBL19732194 0.76 ACHE (0.48) HTTMAPTALDH1A1KMT2ATSHR
SCHEMBL10325884 0.76 HTT (0.51) ERN1HTTMAPTALDH1A1PKM
SCHEMBL8334546 0.75 KMT2A (0.52) ERN1HTTMAPTALDH1A1PKM
SCHEMBL21582162 0.75 TSHR (0.45) HTTALDH1A1KMT2ATSHRAPOBEC3A
SCHEMBL21582165 0.75 TSHR (0.49) HTTALDH1A1TSHRAPOBEC3AAPOBEC3G

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3938350-A1 3-(2-BROM-4-ALKYNYL-6-ALKOXYPHENYL)-SUBSTITUTED 5-SPIROCYCLOHEXYL-3-PYRROLIN-2-ONES AND THEIR USE AS HERBICIDES Bayer Aktiengesellschaft (DE) 2022-01-19 EP disclosed
EP-3938348-A1 NOVEL 3-(2-BROM-4-ALKYNYL-6-ALKOXYPHENYL)-3-PYRROLIN-2-ONES AND THEIR USE AS HERBICIDES Bayer Aktiengesellschaft (DE) 2022-01-19 EP disclosed
CN-113557231-A Novel 3- (2-bromo-4-alkynyl-6-alkoxyphenyl) -3-pyrrolin-2-ones and their use as herbicides 拜耳公司 2021-10-26 CN disclosed
CN-113544119-A 3- (2-bromo-4-alkynyl-6-alkoxyphenyl) -substituted 5-spirocyclohexyl-3-pyrrolin-2-ones and their use as herbicides 拜耳公司 2021-10-22 CN disclosed
EP-3793977-A1 2-BROMO-6-ALKOXYPHENYL-SUBSTITUTED PYRROLIN-2-ONES AND THEIR USE AS HERBICIDES Bayer Aktiengesellschaft (DE) 2021-03-24 EP disclosed
CN-112334446-A 2-bromo-6-alkoxyphenyl-substituted pyrrolin-2-ones and their use as herbicides 拜耳公司 2021-02-05 CN disclosed
WO-2020187627-A1 NOVEL 3-(2-BROM-4-ALKYNYL-6-ALKOXYPHENYL)-3-PYRROLIN-2-ONES AND THEIR USE AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2020-09-24 WO disclosed
WO-2020187629-A1 3-(2-BROM-4-ALKYNYL-6-ALKOXYPHENYL)-SUBSTITUTED 5-SPIROCYCLOHEXYL-3-PYRROLIN-2-ONES AND THEIR USE AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2020-09-24 WO disclosed
WO-2019228788-A1 2-BROMO-6-ALKOXYPHENYL-SUBSTITUTED PYRROLIN-2-ONES AND THEIR USE AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 2019-12-05 WO disclosed