SCHEMBL21584428

SCHEMBL21584428

COc1c(Cl)ccc(-c2nc(NCc3ncccc3C)c(Cl)c(C(=O)OCc3ccccc3)n2)c1F

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.38
NPSR1 Q6W5P4 2/20 0.35
GAA P10253 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
PDE5A O76074 3/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
ADORA2A P29274 3/20 0.34
ADORA1 P30542 2/20 0.34
PDE10A Q9Y233 1/20 0.34
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21584408 0.84 LMNA (0.43) POLBNPSR1GAACYP1A2CYP3A4
SCHEMBL21584389 0.84 CYP1A2 (0.36) POLBNPSR1GAACYP1A2CYP3A4
SCHEMBL21584477 0.83 ALDH1A1 (0.41) POLBGAAMEN1ALDH1A1MAPT
SCHEMBL21584404 0.83 CYP1A2 (0.36) NPSR1GAACYP1A2CYP3A4CYP2C9
SCHEMBL21584461 0.82 KDM4E (0.40) POLBNPSR1GAACYP2C9CYP2C19
SCHEMBL21584416 0.82 ACP1 (0.35) POLBGAACYP1A2MEN1ALDH1A1
SCHEMBL1654721 0.82 CYP1A2 (0.43) POLBNPSR1GAACYP1A2CYP3A4
SCHEMBL2683282 0.80 ADORA2A (0.35) ADORA2AADORA1
SCHEMBL21584377 0.80 GAA (0.38) POLBGAAALDH1A1KMT2ATSHR
SCHEMBL21584335 0.78 MAPT (0.40) POLBALDH1A1MAPTKMT2AADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019227771-A1 SUBSTITUTED PYRIMIDINE-4-FORMIC ACID DERIVATIVE, HERBICIDAL COMPOSITION AND USE THEREOF 青岛清原化合物有限公司 (CN) 2019-12-05 WO disclosed