SCHEMBL21588804

SCHEMBL21588804

Cc1nn(CC(F)(F)F)cc1Nc1ncc(Br)c(NCc2ccc(S(C)(=O)=O)cc2)n1

nearest known ligand 0.87

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 6/20 0.87
LRRK2 Q5S007 6/20 0.87
MKNK2 Q9HBH9 4/20 0.87
IKBKE Q14164 3/20 0.87
CSF1R P07333 3/20 0.87
ULK3 Q6PHR2 3/20 0.87
AAK1 Q2M2I8 3/20 0.87
NUAK2 Q9H093 2/20 0.87
STK17B O94768 1/20 0.87
PI4KB Q9UBF8 1/20 0.87
MARK4 Q96L34 2/20 0.57
STK17A Q9UEE5 2/20 0.55
PTK2 Q05397 5/20 0.47
MYLK2 Q9H1R3 2/20 0.43
NIM1K Q8IY84 1/20 0.43
CYP1A2 P05177 2/20 0.42
NUAK1 O60285 2/20 0.41
STK16 O75716 2/20 0.41
NTRK1 P04629 2/20 0.41
CSNK2A2 P19784 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29710773 0.93 TBK1 (1.00) TBK1LRRK2MKNK2IKBKECSF1R
SCHEMBL21588805 0.93 TBK1 (1.00) TBK1LRRK2MKNK2IKBKECSF1R
SCHEMBL21588811 0.91 LRRK2 (0.73) TBK1LRRK2MKNK2IKBKECSF1R
SCHEMBL21588800 0.85 LRRK2 (0.85) TBK1LRRK2MKNK2IKBKECSF1R
SCHEMBL21588977 0.84 LRRK2 (0.84) TBK1LRRK2MKNK2IKBKECSF1R
SCHEMBL21588815 0.84 LRRK2 (0.83) TBK1LRRK2MKNK2IKBKECSF1R
SCHEMBL21588798 0.84 TBK1 (0.83) TBK1LRRK2MKNK2IKBKECSF1R
SCHEMBL21588799 0.84 LRRK2 (0.83) TBK1LRRK2MKNK2IKBKECSF1R
SCHEMBL21588801 0.82 LRRK2 (0.80) TBK1LRRK2MKNK2IKBKECSF1R
SCHEMBL21588827 0.82 TBK1 (0.79) TBK1LRRK2MKNK2IKBKECSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019233891-A1 TBK1 INHIBITOR COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-12-12 WO disclosed