SCHEMBL21590187

SCHEMBL21590187

CN1CCN(c2ccc([N+](=O)[O-])cc2C2CC2)CC1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.54
LMNA P02545 4/20 0.54
GAA P10253 2/20 0.54
SIRT6 Q8N6T7 1/20 0.54
KMT2A Q03164 3/20 0.52
HTT P42858 3/20 0.52
CYP1A2 P05177 2/20 0.52
CYP3A4 P08684 2/20 0.52
CYP2C19 P33261 2/20 0.52
MEN1 O00255 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.51
WDR5 P61964 4/20 0.51
POLB P06746 2/20 0.51
KDM4E B2RXH2 1/20 0.50
HSP90AA1 P07900 1/20 0.49
HIF1A Q16665 1/20 0.48
MCL1 Q07820 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24630259 0.83 ALDH1A1 (0.65) ALDH1A1LMNAKMT2AHTTCYP1A2
SCHEMBL398803 0.80 ALDH1A1 (0.61) ALDH1A1LMNAGAASIRT6KMT2A
SCHEMBL30464734 0.80 ALDH1A1 (0.66) ALDH1A1LMNAGAASIRT6KMT2A
SCHEMBL3313887 0.80 GAA (0.72) ALDH1A1LMNAGAASIRT6KMT2A
SCHEMBL2461666 0.80 ALDH1A1 (0.66) ALDH1A1LMNAGAASIRT6KMT2A
SCHEMBL15961236 0.80 SIRT6 (0.59) ALDH1A1LMNAGAASIRT6KMT2A
SCHEMBL30410222 0.80 ALDH1A1 (0.61) ALDH1A1LMNAGAASIRT6KMT2A
SCHEMBL1969786 0.79 ALDH1A1 (0.71) ALDH1A1LMNAGAASIRT6KMT2A
SCHEMBL6830223 0.78 ALDH1A1 (0.62) ALDH1A1LMNAGAASIRT6KMT2A
SCHEMBL283385 0.78 SIRT6 (0.58) ALDH1A1LMNAGAASIRT6KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023011610-A1 BENZODIOXANE COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 南京红云生物科技有限公司 2023-02-09 WO disclosed
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed
WO-2019238067-A1 PYRROLO [2, 3-B] PYRIDINES OR PYRROLO [2, 3-B] PYRAZINES AS HPK1 INHIBITOR AND THE USE THEREOF BEIGENE, LTD. (KY) 2019-12-19 WO disclosed