SCHEMBL21590191

SCHEMBL21590191

COCCN(C)c1cc(Br)ccc1[N+](=O)[O-]

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
KDM4E B2RXH2 2/20 0.46
VCAM1 P19320 1/20 0.42
HCAR3 P49019 2/20 0.39
LMNA P02545 1/20 0.38
MAPT P10636 7/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
ABCB1 P08183 1/20 0.36
ABCC1 P33527 1/20 0.36
PKM P14618 1/20 0.35
HTT P42858 1/20 0.35
S100A4 P26447 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
GAA P10253 2/20 0.34
CYP19A1 P11511 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29833175 0.83 ALDH1A1 (0.46) ALDH1A1KDM4EVCAM1HCAR3LMNA
SCHEMBL15616427 0.83 ALDH1A1 (0.48) ALDH1A1KDM4EVCAM1HCAR3MAPT
SCHEMBL18228017 0.81 ALDH1A1 (0.46) ALDH1A1KDM4EVCAM1HCAR3LMNA
SCHEMBL34467410 0.80 HCAR3 (0.47) ALDH1A1KDM4EVCAM1HCAR3LMNA
SCHEMBL21590304 0.80 ALDH1A1 (0.45) ALDH1A1KDM4EVCAM1HCAR3LMNA
SCHEMBL15111028 0.79 ALDH1A1 (0.38) ALDH1A1KDM4EVCAM1HCAR3LMNA
SCHEMBL18508188 0.78 HCAR3 (0.39) ALDH1A1KDM4EVCAM1HCAR3LMNA
SCHEMBL18508297 0.78 HCAR3 (0.39) ALDH1A1KDM4EVCAM1HCAR3LMNA
SCHEMBL1844442 0.77 MAPT (0.47) ALDH1A1KDM4EHCAR3LMNAMAPT
SCHEMBL6541812 0.76 KMT2A (0.46) ALDH1A1KDM4EHCAR3MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112243439-A Pyrrolo [2,3-B ] pyridines or pyrrolo [2,3-B ] pyrazines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-01-19 CN disclosed
WO-2019238067-A1 PYRROLO [2, 3-B] PYRIDINES OR PYRROLO [2, 3-B] PYRAZINES AS HPK1 INHIBITOR AND THE USE THEREOF BEIGENE, LTD. (KY) 2019-12-19 WO disclosed