SCHEMBL21590280

SCHEMBL21590280

COc1cc(Cl)ccc1C1CCCCN1C

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
MAPK1 P28482 1/20 0.44
KDM4E B2RXH2 1/20 0.42
POLB P06746 1/20 0.42
HPGD P15428 1/20 0.42
RAB9A P51151 1/20 0.42
GAA P10253 1/20 0.41
TSHR P16473 1/20 0.41
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
HTR3A P46098 1/20 0.40
HTR3D Q70Z44 1/20 0.40
HTR3C Q8WXA8 1/20 0.40
GRM5 P41594 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21590273 0.83 KDM4E (0.46) KDM4EGAA
SCHEMBL13634928 0.79 MEN1 (0.51) ALDH1A1
SCHEMBL16457216 0.77 GAA (0.47) GAATSHR
SCHEMBL11629932 0.75 GAA (0.48) ALDH1A1POLBGAATSHR
SCHEMBL22062939 0.75 MEN1 (0.51) HTR3A
SCHEMBL7031252 0.74 HTR2A (0.44) ALDH1A1MAPK1KDM4E
SCHEMBL13162085 0.74 CHRNB4 (0.54) ALDH1A1
SCHEMBL28973912 0.74 CHRNB2 (0.46)
SCHEMBL4572970 0.73 PTGDR2 (0.49) TSHR
SCHEMBL4573099 0.73 MEN1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019238067-A1 PYRROLO [2, 3-B] PYRIDINES OR PYRROLO [2, 3-B] PYRAZINES AS HPK1 INHIBITOR AND THE USE THEREOF BEIGENE, LTD. (KY) 2019-12-19 WO disclosed