SCHEMBL21593337

SCHEMBL21593337

Cc1onc(-c2ccc(Cl)nc2)c1Cn1ncc(N2CC[C@@H]2C)cc1=O

nearest known ligand 0.39

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 16/20 0.39
ALDH1A1 P00352 1/20 0.34
GABRA5 P31644 1/20 0.33
TAS2R8 Q9NYW2 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30694896 0.87 GABRA1 (0.38) GABRA1GABRA5TAS2R8
SCHEMBL23150882 0.87 GABRA1 (0.38) GABRA1GABRA5TAS2R8
SCHEMBL21590977 0.87 GABRA1 (0.38) GABRA1GABRA5TAS2R8
SCHEMBL30694841 0.87 GABRA1 (0.38) GABRA1GABRA5TAS2R8
SCHEMBL30694843 0.85 GABRA1 (0.37) GABRA1GABRA5
SCHEMBL21590900 0.85 GABRA1 (0.37) GABRA1GABRA5
SCHEMBL21590573 0.85 GABRA1 (0.37) GABRA1ALDH1A1GABRA5
SCHEMBL21593268 0.85 GABRA1 (0.37) GABRA1ALDH1A1GABRA5
SCHEMBL21593336 0.84 GABRA1 (0.39) GABRA1
SCHEMBL21590915 0.84 GABRA1 (0.36) GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019238633-A1 NEW ISOXAZOLYL ETHER DERIVATIVES AS GABA A ALPHA5 PAM F. HOFFMANN-LA ROCHE AG (CH) 2019-12-19 WO disclosed