SCHEMBL21595889

SCHEMBL21595889

COc1cc(Cl)ccc1OCCN(C)C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.54
GAA P10253 1/20 0.54
MAPK1 P28482 1/20 0.54
ALDH1A1 P00352 5/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
MRGPRX4 Q96LA9 1/20 0.47
PTGES O14684 1/20 0.46
S1PR4 O95977 1/20 0.45
FLT3 P36888 1/20 0.45
PSEN1 P49768 1/20 0.45
PSEN2 P49810 1/20 0.45
APH1B Q8WW43 1/20 0.45
NCSTN Q92542 1/20 0.45
APH1A Q96BI3 1/20 0.45
PSENEN Q9NZ42 1/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
LMNA P02545 1/20 0.45
TDP1 Q9NUW8 1/20 0.44
FDPS P14324 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21596090 0.86 KDM4E (0.56) KDM4EGAAMAPK1ALDH1A1SMN1; SMN2
SCHEMBL21595706 0.84 KDM4E (0.56) KDM4EGAAMAPK1ALDH1A1SMN1; SMN2
SCHEMBL21595924 0.83 KDM4E (0.54) KDM4EGAAMAPK1ALDH1A1SMN1; SMN2
SCHEMBL21596073 0.83 ALDH1A1 (0.48) KDM4EALDH1A1MEN1KMT2ALMNA
SCHEMBL21601500 0.83 KDM4E (0.49) KDM4EGAAMAPK1ALDH1A1SMN1; SMN2
SCHEMBL27164592 0.81 FDPS (0.67) KDM4EALDH1A1SMN1; SMN2LMNAFDPS
SCHEMBL9799953 0.78 MAPT (0.61) KDM4EALDH1A1SMN1; SMN2PTGESMEN1
SCHEMBL1332214 0.76 TDP1 (0.68) KDM4ESMN1; SMN2MEN1KMT2ATDP1
SCHEMBL21595882 0.76 HRH3 (0.58) KDM4EALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL21595943 0.76 ALDH1A1 (0.54) KDM4EALDH1A1SMN1; SMN2MRGPRX4S1PR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019244066-A2 PYRIDIN-3-YL ACETIC ACID DERIVATIVES AS INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV Healthcare UK (No.5) Limited (GB) 2019-12-26 WO disclosed