SCHEMBL21595952

SCHEMBL21595952

Cc1ccc(OCCN(C)C(=O)O)c(Cl)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 11/20 0.68
MAPT P10636 5/20 0.56
MAPK1 P28482 4/20 0.56
ATM Q13315 3/20 0.56
ALDH1A1 P00352 7/20 0.55
TDP1 Q9NUW8 3/20 0.55
LMNA P02545 1/20 0.55
PPARG P37231 1/20 0.52
GAA P10253 2/20 0.51
MRGPRX4 Q96LA9 1/20 0.49
L3MBTL1 Q9Y468 3/20 0.49
RAB9A P51151 2/20 0.49
NPBWR1 P48145 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MCHR1 Q99705 1/20 0.47
NPY1R P25929 1/20 0.46
NPY2R P49146 1/20 0.46
HPGD P15428 2/20 0.46
NPC1 O15118 1/20 0.46
KMT2A Q03164 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16585308 0.87 KDM4E (0.72) KDM4EMAPTALDH1A1TDP1LMNA
SCHEMBL21596090 0.87 KDM4E (0.56) KDM4EMAPTMAPK1ALDH1A1TDP1
SCHEMBL21595725 0.85 KDM4E (0.54) KDM4EMAPTMAPK1ATMALDH1A1
SCHEMBL21595734 0.84 KDM4E (0.51) KDM4EMAPTMAPK1ATMALDH1A1
SCHEMBL21601488 0.83 KDM4E (0.55) KDM4EMAPTMAPK1ATMALDH1A1
SCHEMBL10828209 0.81 KDM4E (0.49) KDM4EMAPTMAPK1ATMALDH1A1
SCHEMBL9158338 0.80 LTA4H (0.53) KDM4EMAPTMAPK1ATMALDH1A1
SCHEMBL21595706 0.80 KDM4E (0.56) KDM4EMAPK1ALDH1A1TDP1GAA
SCHEMBL10359783 0.79 PPARG (0.67) KDM4EMAPTMAPK1ATMALDH1A1
SCHEMBL15445592 0.79 TSHR (0.71) KDM4EMAPTMAPK1ATMALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019244066-A2 PYRIDIN-3-YL ACETIC ACID DERIVATIVES AS INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV Healthcare UK (No.5) Limited (GB) 2019-12-26 WO disclosed