SCHEMBL21596337

SCHEMBL21596337

NC(=O)c1cnc(Cl)nc1Oc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 5/20 0.55
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
TDP1 Q9NUW8 2/20 0.50
RAB9A P51151 1/20 0.49
CTNNB1 P35222 1/20 0.47
POLB P06746 3/20 0.45
CYP1A2 P05177 3/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
ALDH1A1 P00352 1/20 0.43
PARP10 Q53GL7 1/20 0.42
BTK Q06187 1/20 0.42
SYK P43405 1/20 0.42
CASP6 P55212 1/20 0.42
PLA2G10 O15496 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16670419 0.97 PIN1 (0.52) PIN1MEN1KMT2ATDP1RAB9A
SCHEMBL26984449 0.83 TDP1 (0.58) PIN1MEN1KMT2ATDP1RAB9A
SCHEMBL16597748 0.81 SCN9A (0.54) PIN1MEN1KMT2ATDP1RAB9A
SCHEMBL13919652 0.81 XPO1 (0.60) PIN1MEN1KMT2ATDP1ALDH1A1
SCHEMBL17673007 0.80 PIN1 (0.56) PIN1POLBPARP10
SCHEMBL26984232 0.80 CYP1A2 (0.72) PIN1MEN1KMT2ATDP1RAB9A
SCHEMBL29193018 0.79 RAB9A (0.51) MEN1KMT2ATDP1RAB9ACTNNB1
SCHEMBL16670315 0.77 KMT2A (0.50) MEN1KMT2ATDP1CTNNB1POLB
SCHEMBL16670718 0.77 BTK (0.53) MEN1KMT2ATDP1RAB9ACTNNB1
SCHEMBL12620334 0.76 PIN1 (0.60) PIN1MEN1KMT2ARAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112313207-B Cyano-substituted pyridine and cyano-substituted pyrimidine compounds, and preparation methods and applications thereof 北京赛特明强医药科技有限公司 2023-02-14 CN disclosed
CN-112313207-A Cyano-substituted pyridine and cyano-substituted pyrimidine compounds, and preparation methods and applications thereof 北京赛特明强医药科技有限公司 2021-02-02 CN disclosed
WO-2019242689-A1 CYANO-SUBSTITUTED PYRIDINE AND CYANO-SUBSTITUTED PYRIMIDINE COMPOUND, AND PREPARATION METHOD AND APPLICATION THEREOF 北京赛特明强医药科技有限公司 2019-12-26 WO disclosed
WO-2019242689-A1 CYANO-SUBSTITUTED PYRIDINE AND CYANO-SUBSTITUTED PYRIMIDINE COMPOUND, AND PREPARATION METHOD AND APPLICATION THEREOF 北京赛特明强医药科技有限公司 2019-12-26 WO disclosed