SCHEMBL21600577

SCHEMBL21600577

OCc1c[nH]c2c(F)ccc(Br)c12

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.43
GPR84 Q9NQS5 4/20 0.42
MPO P05164 7/20 0.39
SLC6A4 P31645 5/20 0.39
RIPK1 Q13546 1/20 0.33
FFAR1 O14842 1/20 0.32
PCSK9 Q8NBP7 2/20 0.31
TNF P01375 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5387311 0.87 HTR1A (0.48) HTR1AGPR84MPOSLC6A4
SCHEMBL5398443 0.80 HTR1A (0.42) HTR1AGPR84MPOSLC6A4TNF
SCHEMBL5392766 0.79 HTR1A (0.38) HTR1AGPR84MPOSLC6A4RIPK1
SCHEMBL30457622 0.73 HTR1A (0.33) HTR1AGPR84
SCHEMBL20576934 0.73 ALDH1A1 (0.35) HTR1AGPR84RIPK1TNF
SCHEMBL19216724 0.73 HTR1A (0.36) HTR1AGPR84
SCHEMBL14663023 0.69 CYP2A6 (0.51) HTR1A
SCHEMBL31663177 0.69 HTR2A (0.32)
SCHEMBL29953964 0.69 CYP2A6 (0.51) HTR1A
SCHEMBL25381397 0.68 CYP2A6 (0.50) HTR1AGPR84FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3202766-B1 ISOXAZOLE DERIVATIVE AS MUTATED ISOCITRATE DEHYDROGENASE 1 INHIBITOR DAIICHI SANKYO CO LTD (JP) 2019-12-25 EP disclosed