SCHEMBL21603015

SCHEMBL21603015

C(#Cc1ccn(-c2ccccc2)c1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.50
COMT P21964 1/20 0.44
MAPT P10636 2/20 0.40
GRM5 P41594 5/20 0.38
DRD4 P21917 2/20 0.38
CYP3A4 P08684 3/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.36
KCNH2 Q12809 1/20 0.35
THPO P40225 1/20 0.34
CA12 O43570 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19454389 0.87 APP (0.41) APPCOMTMAPTGRM5MEN1
SCHEMBL8772892 0.79 GRM5 (0.48) COMTGRM5DRD4CYP3A4
SCHEMBL402534 0.74 APP (0.55) APPMAPTGRM5CYP3A4CYP1A2
Diphenylacetylene SCHEMBL960609 0.71 APP (1.00) APPMAPTGRM5CYP3A4CYP1A2
Diphenylacetylene SCHEMBL68254 0.71 APP (1.00) APPMAPTGRM5CYP3A4CYP1A2
Diphenylacetylene SCHEMBL29188592 0.71 APP (1.00) APPMAPTGRM5CYP3A4CYP1A2
Diphenylacetylene SCHEMBL23754282 0.68 APP (0.92) APPMAPTGRM5CYP3A4CYP1A2
Diphenylacetylene SCHEMBL31286315 0.68 APP (0.92) APPMAPTGRM5CYP3A4CYP1A2
Diphenylacetylene SCHEMBL9273707 0.68 APP (0.92) APPMAPTGRM5CYP3A4CYP1A2
Diphenylacetylene SCHEMBL31243352 0.68 APP (0.92) APPMAPTGRM5CYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3810571-A1 COMPOUNDS FOR THE TREATMENT OF BOVINE OR SWINE RESPIRATORY DISEASE Intervet International B.V. (NL) 2021-04-28 EP disclosed
WO-2020002238-A1 COMPOUNDS FOR THE TREATMENT OF BOVINE OR SWINE RESPIRATORY DISEASE INTERVET INTERNATIONAL B.V. (NL) 2020-01-02 WO disclosed