SCHEMBL21616752

SCHEMBL21616752

C=Cc1ccc(CO)c(OC)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.61
PDCD1 Q15116 1/20 0.46
CD274 Q9NZQ7 1/20 0.46
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
MMP9 P14780 3/20 0.43
MMP2 P08253 2/20 0.43
MMP8 P22894 2/20 0.43
NFKB1 P19838 2/20 0.43
ALDH1A1 P00352 3/20 0.40
HPGD P15428 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
TRIM24 O15164 1/20 0.40
ALDH5A1 P51649 1/20 0.40
ABAT P80404 1/20 0.40
TRIM33 Q9UPN9 1/20 0.40
NFE2L2 Q16236 2/20 0.39
TSHR P16473 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14107081 0.84 TRPA1 (0.58) TRPA1MMP9NFKB1ALDH1A1HPGD
SCHEMBL810242 0.82 TRPA1 (0.56) TRPA1ALDH1A1HPGDTDP1TRIM24
SCHEMBL14761112 0.82 TRPA1 (0.56) TRPA1ALDH1A1HPGDTDP1TRIM24
SCHEMBL10031796 0.82 ALDH1A1 (0.61) PDCD1CD274MMP9MMP2MMP8
SCHEMBL16950361 0.81 TRPA1 (0.54) TRPA1ALDH1A1TSHRPTGS1PTGS2
SCHEMBL14760865 0.79 TRPA1 (0.53) TRPA1ALDH1A1HPGDTDP1TRIM24
SCHEMBL15524839 0.79 TRPA1 (0.53) TRPA1ALDH1A1TSHRGAAMAPT
SCHEMBL12233281 0.79 PDCD1 (0.44) TRPA1PDCD1CD274PDE4APDE4B
SCHEMBL27377995 0.78 APP (0.41) TRPA1ALDH1A1HPGDAPP
SCHEMBL26874268 0.77 TRPA1 (0.46) TRPA1PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111886219-B Immunosuppressant, preparation method and pharmaceutical application thereof 上海和誉生物医药科技有限公司 2023-04-25 CN disclosed
CN-111886219-A Immunosuppressant, preparation method and pharmaceutical application thereof 上海和誉生物医药科技有限公司 2020-11-03 CN disclosed
WO-2020011209-A1 IMMUNOSUPPRESSIVE AGENT, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USE THEREOF 上海和誉生物医药科技有限公司 2020-01-16 WO disclosed
WO-2020011209-A1 IMMUNOSUPPRESSIVE AGENT, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USE THEREOF 上海和誉生物医药科技有限公司 2020-01-16 WO disclosed