SCHEMBL21620194

SCHEMBL21620194

O=Cc1cnc(N2CCC(c3ccc(C(F)(F)F)cc3)C2)nc1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.43
AOC3 Q16853 1/20 0.41
SCN10A Q9Y5Y9 1/20 0.41
CYP3A4 P08684 2/20 0.41
SLC6A9 P48067 6/20 0.39
PROKR1 Q8TCW9 2/20 0.39
HTR2C P28335 1/20 0.38
MCHR1 Q99705 1/20 0.37
NOTUM Q6P988 1/20 0.37
GRM2 Q14416 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21620073 0.86 KDM4E (0.46) ACACBAOC3SCN10ACYP3A4SLC6A9
SCHEMBL21619819 0.85 ACACB (0.46) ACACBAOC3SCN10ACYP3A4SLC6A9
SCHEMBL21616612 0.84 CYP3A4 (0.43) ACACBAOC3SCN10ACYP3A4SLC6A9
SCHEMBL28539978 0.81 ACACB (0.41) ACACBAOC3SCN10ACYP3A4SLC6A9
SCHEMBL23636875 0.80 LIPG (0.49) ACACB
SCHEMBL17832257 0.77 SCN9A (0.44) MCHR1GRM2
SCHEMBL17832258 0.77 DHFR (0.48) CYP3A4
SCHEMBL21619936 0.74 ACACB (0.38) ACACBPROKR1HTR2C
SCHEMBL17832213 0.74 OGA (0.43) AOC3
SCHEMBL21620016 0.74 TRIM24 (0.48) PROKR1HTR2CNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020011147-A1 RORγ ANTAGONIST AND APPLICATION THEREOF IN MEDICINE SUNSHINE LAKE PHARMA CO., LTD. (CN) 2020-01-16 WO disclosed