SCHEMBL21622374

SCHEMBL21622374

CN1Cc2cc(Br)cnc2C1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABHD6 Q9BV23 1/20 0.44
HSD17B10 Q99714 1/20 0.38
HRH4 Q9H3N8 2/20 0.34
HRH3 Q9Y5N1 2/20 0.34
HTT P42858 2/20 0.33
KMT2A Q03164 1/20 0.33
CYP2C19 P33261 1/20 0.32
BRD4 O60885 1/20 0.32
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8022098 0.85 CYP2C19 (0.44) ABHD6HSD17B10KMT2ACYP2C19MAPT
SCHEMBL30033295 0.85 CYP2C19 (0.44) ABHD6HSD17B10KMT2ACYP2C19MAPT
SCHEMBL25690672 0.78 ABHD6 (0.47) ABHD6HSD17B10HTTKMT2A
SCHEMBL14881091 0.78 ABHD6 (0.47) ABHD6HSD17B10HTTKMT2ASMN1; SMN2
SCHEMBL14907172 0.78 CCR1 (0.34) HRH4CYP2C19CYP2C9
SCHEMBL19080449 0.76 SLC6A2 (0.34) ABHD6CYP2C19SMN1; SMN2CYP2C9
SCHEMBL21937114 0.75 ABHD6 (0.42) ABHD6HTTCYP2C19MAPT
SCHEMBL21802762 0.75 ABHD6 (0.58) ABHD6HTTKMT2ASMN1; SMN2ALDH1A1
SCHEMBL12341045 0.73 HPGD (0.34) ABHD6HRH3HTTCYP2C19BRD4
SCHEMBL12344128 0.73 HRH3 (0.40) HRH4HRH3CYP2C19MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3822266-A1 PYRROLIDINYL UREA DERIVATIVES AND APPLICATION THEREOF IN TRKA-RELATED DISEASES Zhangzhou Pien Tze Huang Pharmaceutical Co., Ltd (CN) 2021-05-19 EP disclosed
WO-2020083377-A1 PYRROLIDINYL UREA DERIVATIVES AND APPLICATION THEREOF 南京明德新药研发有限公司 2020-04-30 WO disclosed
WO-2020011227-A1 PYRROLIDINYL UREA DERIVATIVES AND APPLICATION THEREOF IN TRKA-RELATED DISEASES 南京明德新药研发有限公司 2020-01-16 WO disclosed