SCHEMBL2164206

SCHEMBL2164206

CC(C)(C)OC(=O)NCCC(=O)c1cccc(N(CCc2ccccc2)C(=O)OC(C)(C)C)c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.44
IDO1 P14902 1/20 0.41
NQO2 P16083 1/20 0.39
CTSK P43235 2/20 0.39
CTSS P25774 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
POLB P06746 1/20 0.38
KDM4E B2RXH2 1/20 0.37
NAMPT P43490 1/20 0.37
NR1H4 Q96RI1 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37
CKS1B P61024 1/20 0.37
SKP1 P63208 1/20 0.37
SKP2 Q13309 1/20 0.37
PTPN1 P18031 1/20 0.36
F2 P00734 1/20 0.36
DRD2 P14416 1/20 0.36
AKT1 P31749 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2779187 0.93 SIGMAR1 (0.45) SIGMAR1IDO1NQO2CTSKCTSS
SCHEMBL2168456 0.90 NR1H4 (0.44) SIGMAR1IDO1NQO2CTSSNPSR1
SCHEMBL2151042 0.88 SIGMAR1 (0.48) SIGMAR1IDO1CTSKNPSR1POLB
SCHEMBL2164881 0.86 NR1H4 (0.45) SIGMAR1IDO1CTSSNR1H4TMEM97
SCHEMBL3138728 0.79 L3MBTL1 (0.48) SIGMAR1IDO1CTSSNPSR1NR1H4
SCHEMBL3134720 0.79 EPHX1 (0.39) NQO2KDM4ENR1H4
SCHEMBL2164212 0.78 ACE (0.42) SIGMAR1IDO1CTSKCTSSTMEM97
SCHEMBL3135260 0.77 HDAC1 (0.37) SIGMAR1IDO1POLBKDM4ENR1H4
SCHEMBL942893 0.77 IDO1 (0.51) SIGMAR1IDO1KDM4ECKS1BSKP1
SCHEMBL2150723 0.76 ACACB (0.40) SIGMAR1NQO2KDM4ENR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2340242-A2 COMPOUNDS FOR TREATING OPHTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2011-07-06 EP disclosed