SCHEMBL21644512

SCHEMBL21644512

CC(C)c1cc(C(=O)Nc2ccncc2)c(O)cc1O

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.59
RAB9A P51151 1/20 0.59
KCNMA1 Q12791 2/20 0.56
BCL2 P10415 1/20 0.51
TYK2 P29597 7/20 0.49
JAK2 O60674 5/20 0.47
JAK1 P23458 2/20 0.47
KDM4E B2RXH2 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
ROCK2 O75116 3/20 0.46
ROCK1 Q13464 3/20 0.46
HTT P42858 1/20 0.46
PRKAB2 O43741 1/20 0.45
PRKAG1 P54619 1/20 0.45
PRKAA2 P54646 1/20 0.45
PRKAA1 Q13131 1/20 0.45
PRKAG3 Q9UGI9 1/20 0.45
PRKAG2 Q9UGJ0 1/20 0.45
PRKAB1 Q9Y478 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21644634 0.85 BCL2 (0.69) NPC1RAB9ABCL2KDM4EHTT
SCHEMBL21644571 0.84 KCNMA1 (0.60) NPC1RAB9AKCNMA1BCL2KDM4E
SCHEMBL21644546 0.83 P2RX1 (0.56) NPC1RAB9ABCL2KDM4EHTT
SCHEMBL21644609 0.77 SMN1; SMN2 (0.54) NPC1RAB9ABCL2HTT
SCHEMBL21644596 0.76 NPC1 (0.58) NPC1RAB9AHTT
SCHEMBL30474350 0.75 HSP90AA1 (0.56) BCL2
SCHEMBL21644578 0.75 ALDH1A1 (0.59) NPC1RAB9AHTT
SCHEMBL21644539 0.75 TMPRSS4 (0.63) NPC1RAB9AKDM4EL3MBTL1
SCHEMBL15478027 0.75 NPC1 (1.00) NPC1RAB9AKCNMA1KDM4E
SCHEMBL28421724 0.74 TYK2 (0.56) TYK2JAK2JAK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111164074-B Heat shock protein 90 inhibitors 台北医学大学 2024-02-02 CN disclosed
US-11479528-B2 Heat shock protein 90 inhibitors TAIPEI MEDICAL UNIVERSITY (TW) 2022-10-25 US disclosed
CN-111164074-A Heat shock protein 90 inhibitor 台北医学大学 2020-05-15 CN disclosed
US-20200039923-A1 HEAT SHOCK PROTEIN 90 INHIBITORS TAIPEI MEDICAL UNIVERSITY (TW) 2020-02-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200039923-A1 HEAT SHOCK PROTEIN 90 INHIBITORS HSP90AB1, HSP90AB2P, HSP90AA1 NPC1 1353/4885RAB9A 1972/4885KCNMA1 4571/4885
US-11479528-B2 Heat shock protein 90 inhibitors HSP90AB1, HSP90AB2P, HSP90AA1 NPC1 1353/4885RAB9A 1972/4885KCNMA1 4571/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.